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CB1R antagonist 1

🥰Excellent
Catalog No. T61989Cas No. 334668-69-8

CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.

CB1R antagonist 1

CB1R antagonist 1

🥰Excellent
Purity: 99.65%
Catalog No. T61989Cas No. 334668-69-8
CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.
Pack SizePriceAvailabilityQuantity
5 mg64 €In Stock
10 mg112 €In Stock
25 mg188 €In Stock
50 mg278 €In Stock
100 mg416 €In Stock
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Purity:99.65%
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Product Introduction

Bioactivity
Description
CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.
Targets&IC50
CB1 receptor (human):4.2 uM, CB1 receptor (human):10 uM (EC50)
In vitro
CB1R antagonist 1 exhibits cannabinoid-1 receptor (CB1R) activity with an IC50 value of 4.2 μM and an EC50 value greater than 10 μM [1].
Chemical Properties
Molecular Weight404.45
FormulaC18H23F3N2O3S
Cas No.334668-69-8
SmilesS(=O)(=O)(C1=CC(C(F)(F)F)=CC=C1)N2CCN(C(=O)C3CCCCC3)CC2
Storage & Solubility Information
StorageShipping with blue ice.
Solubility Information
DMSO: 80 mg/mL (197.80 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4725 mL12.3625 mL24.7249 mL123.6247 mL
5 mM0.4945 mL2.4725 mL4.9450 mL24.7249 mL
10 mM0.2472 mL1.2362 mL2.4725 mL12.3625 mL
20 mM0.1236 mL0.6181 mL1.2362 mL6.1812 mL
50 mM0.0494 mL0.2472 mL0.4945 mL2.4725 mL
100 mM0.0247 mL0.1236 mL0.2472 mL1.2362 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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