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CFTR corrector 8
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CFTR corrector 8
Catalog No. T63806Cas No. 1918142-35-4
CFTR corrector 8 is a highly effective modulator of the cystic fibrosis transmembrane conductance regulator (CFTR). This compound is specifically designed for utilization in research related to cystic fibrosis, a genetic disorder primarily affecting the lungs and digestive system [1].
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $272 | In Stock | |
| 5 mg | $677 | In Stock | |
| 10 mg | $963 | In Stock | |
| 25 mg | $1,430 | In Stock | |
| 50 mg | $1,930 | In Stock | |
| 100 mg | $2,590 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $987 | In Stock |
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CFTR corrector 4
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | CFTR corrector 8 is a highly effective modulator of the cystic fibrosis transmembrane conductance regulator (CFTR). This compound is specifically designed for utilization in research related to cystic fibrosis, a genetic disorder primarily affecting the lungs and digestive system [1]. |
| In vitro | CFTR corrector 8 demonstrates EC50 values of 1 μM in the CSE-HRP assay and 3 μM in the HBE-TECC assay.[1] CFTR corrector 8 displays a hepatocyte clearance rate of 1250 L/hr/kg in humans and 775 L/hr/kg in rats.[1] |
| Molecular Weight | 539.52 |
| Formula | C29H27F2NO7 |
| Cas No. | 1918142-35-4 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||
| Solubility Information | DMSO: 10 mg/mL (18.53 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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