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KI-7
Catalog No. T9238Cas No. 1489263-00-4
KI-7 is an adenosine A2B receptor positive allosteric modulator.
KI-7
Catalog No. T9238Cas No. 1489263-00-4
KI-7 is an adenosine A2B receptor positive allosteric modulator.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $32 | In Stock | |
| 5 mg | $53 | In Stock | |
| 10 mg | $92 | In Stock | |
| 25 mg | $191 | In Stock | |
| 50 mg | $293 | In Stock | |
| 100 mg | $443 | In Stock | |
| 200 mg | $623 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $59 | In Stock |
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CitedSelect Batch
Purity:98.03%
Contact us for more batch information
With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.Product Introduction
Bioactivity
Chemical Properties
| Description | KI-7 is an adenosine A2B receptor positive allosteric modulator. |
| In vitro | KI-7 potentiates the cAMP accumulation induced by the non-selective A2B adenosine receptor agonist NECA (EC50=445.8 nM). KI-7 also potentiates the cAMP accumulation induced by the selective A2B adenosine receptor agonist BAY 60-6583 as well as by adenosine with EC50s of 2390 nM and 2550 nM, respectively[1][2]. |
| Molecular Weight | 354.4 |
| Formula | C23H18N2O2 |
| Cas No. | 1489263-00-4 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 240 mg/mL (677.20 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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