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Lys-Bradykinin acetate(342-10-9 free base)
🥰Excellent
Catalog No. TP2268LCas No. 84640-50-6
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
Lys-Bradykinin acetate(342-10-9 free base)
🥰Excellent
Purity: 99.86%
Catalog No. TP2268LCas No. 84640-50-6
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $98 | In Stock | |
| 5 mg | $223 | In Stock | |
| 10 mg | $333 | In Stock | |
| 25 mg | $563 | In Stock | |
| 50 mg | $792 | In Stock | |
| 100 mg | $1,120 | In Stock | |
| 500 mg | $2,250 | In Stock |
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Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base)
TP1918L1
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. 16-fold more potent than [Des-Arg9]-Bradykinin.
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[Des-Arg9]-Bradykinin acetate is a selective agonist of the Bradykinin B1 receptor.
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Purity:99.86%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist. |
| Molecular Weight | 1248.43 |
| Formula | C58H89N17O14 |
| Cas No. | 84640-50-6 |
| Smiles | NCCCC[C@@H](C(N[C@H](C(N1CCC[C@H]1C(N2CCC[C@H]2C(NCC(N[C@H](C(N[C@H](C(N3CCC[C@H]3C(N[C@H](C(N[C@H](C(O)=O)CCCNC(N)=N)=O)Cc4ccccc4)=O)=O)CO)=O)Cc5ccccc5)=O)=O)=O)=O)CCCNC(N)=N)=O)N.CC(O)=O |
| Relative Density. | 1.31g/cm3 |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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