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N6-(2-Phenylethyl)adenosine
Catalog No. T12163Cas No. 20125-39-7
Alias N6-Phenylethyladenosine, N6-Phenethyladenosine
N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and adenosine receptor agonist with Ki values of 11.8 nM for rat A1 receptors and 30.1 nM for human A1 receptors.
N6-(2-Phenylethyl)adenosine
Catalog No. T12163Alias N6-Phenylethyladenosine, N6-PhenethyladenosineCas No. 20125-39-7
N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and adenosine receptor agonist with Ki values of 11.8 nM for rat A1 receptors and 30.1 nM for human A1 receptors.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $29 | In Stock | |
| 25 mg | $57 | In Stock | |
| 50 mg | $112 | In Stock | |
| 100 mg | $196 | In Stock | |
| 200 mg | $352 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $29 | In Stock |
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CitedSelect Batch
Purity:99.94%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and adenosine receptor agonist with Ki values of 11.8 nM for rat A1 receptors and 30.1 nM for human A1 receptors. |
| Targets&IC50 | A1AR (human):30.1 nM (ki), A1AR (rat):ki:11.8 nM , A3AR (human):0.63 nM (ki) |
| In vitro | The Ki value of human A3 is 0.63 nM. In CHO cells, N6-(2-Phenylethyl)adenosine inhibits A2 with IC50s of 560 nM and 2250 nM for rat and human[1]. |
| Alias | N6-Phenylethyladenosine, N6-Phenethyladenosine |
| Molecular Weight | 371.39 |
| Formula | C18H21N5O4 |
| Cas No. | 20125-39-7 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | H2O: < 0.1 mg/mL (insoluble) DMSO: 95 mg/mL (255.80 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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