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PF-562271 hydrochloride (PF-562271 HCl) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM in cell-free assays, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, except for some CDKs.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | 67 € | In Stock | |
10 mg | 93 € | In Stock | |
25 mg | 147 € | In Stock | |
50 mg | 212 € | In Stock | |
100 mg | 314 € | In Stock |
Description | PF-562271 hydrochloride (PF-562271 HCl) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM in cell-free assays, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, except for some CDKs. |
Targets&IC50 | FAK:1.5 nM |
Alias | PF-562271 HCl |
Molecular Weight | 543.95 |
Formula | C21H20F3N7O3S HCl |
Cas No. | 939791-41-0 |
Smiles | Cl.CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)ncc1C(F)(F)F)S(C)(=O)=O |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 91 mg/mL (167.3 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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