T9552 |
BAZ1A-IN-1
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Epigenetic Reader Domain
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BAZ1A-IN-1 is a potent BAZ1A inhibitor with the KD value of 0.52 μM for the BAZ1A bromodomain. BAZ1A-IN-1 shows good ant... |
T60028 |
MM41
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DNA/RNA Synthesis
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MM41 is a human telomeric and gene promoter DNA quadruplex stabilizer with an IC50 of <10 nM against the MIA PaCa-2 panc... |
TN2064 |
Physcion 8-O-β-D-glucopyranoside
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Physcion 8-O-beta-D-monoglucoside |
TNF
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Physcion 8-O-β-D-glucopyranoside has anti-inflammatory and anti-cancer activities. Physcion 8-O-β-D-glucopyranoside can ... |
T41255 |
SPA70
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Others
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SPA70 is a selective pregnane X receptor (PXR) antagonist with an IC50 of 540 nM and Ki of 390 nM for human PCR and enha... |
T39275 |
Befotertinib
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D-0316 |
EGFR
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Befotertinib is an inhibitor of EGFR tyrosine kinase and can be used for studies about EGFR T790M-positive non-small cel... |
T38815 |
Millepachine
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Apoptosis
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Millepachine is a natural product found in the Chinese herbal medicine with strong antitumor effects against numerous hu... |
T9810 |
TNIK-IN-5
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Wnt/beta-catenin
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TNIK-IN-5 is an potent TNIK inhibitor (IC50= 0.05 μM). TNIK-IN-5 potently inhibits Wnt signaling in intact cells. TNIK-I... |
T60024 |
CFT7455
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CFT7455 is an anti-cancer agent showing high affinity to the cereblon E3 ligase with a Kd of 0.9 nM. CFT7455 is an orall... |
T9882 |
RUVBL1/2 ATPase-IN-1
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Others
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RUVBL1/2 ATPase-IN-1 is an effective RUVBL1/2 ATPase inhibitor with IC50 values of 6.0 and 7.7 μM, respectively. RUVBL1/... |
T39710 |
ARV-471
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Vepdegestrant |
Estrogen Receptor/ERR
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ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the resear... |
T60757 |
SB-216
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SB-216 is able to be used for the research of cancer which is a potent inhibitor of tubulin polymerization. SB-216 exhi... |
T60099 |
RBN013209
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CD38
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RBN013209 is a potent CD38 inhibitor. RBN013209 is useful in the treatment of cancer. |
T41256 |
SP-96
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Aurora Kinase
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SP-96 is a highly effective and selective inhibitor of Aurora B with an IC50 of 0.316 nM. SP-96 shows selective growth i... |
T9912 |
Trastuzumab
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EGFR
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Trastuzumab is a humanized monoclonal antibody for patients with invasive breast cancers that overexpress HER2. Trastuzu... |
T90596 |
Sivifene
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Others
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Sivifene is a antitumor agent. Sivifene can be used for research on the treatment of cutaneous metastases from cancer. |
T8765 |
IGOT1-01
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Others
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iGOT1-01 is an effective inhibitor of glutamate oxaloacetate transaminase 1(GOT1) . iGOT1-01 has IC50s of 84.6 μM and 11... |
T23889 |
CID-663143
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CID663143 |
Microtubule Associated
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CID-663143 inhibits cancer cell growth and shows microtubule-binding activity. |
T9720 |
T3Inh-1
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Others
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T3Inh-1 is an effective and selective inhibitor of ppGalNAc-T3 with an IC50 of 7 µM. T3Inh-1 prevents breast cancer cell... |
T9156 |
CDC25B-IN-2
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Phosphatase
,
mTOR
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BIA is an inhibitor of the interaction between TMBIM6 and mTORC2, which ultimately blocks AKT activation and cancer prog... |
T35329L |
EAD1 HCl
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EAD1 HCL(1644388-26-0 Free base) |
Apoptosis
,
Autophagy
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EAD1 HCL is a potent autophagy inhibitor with antiproliferative activity in lung and pancreatic cancer cells. EAD1 HCL a... |