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Halopemide

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Purity:96.29%

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COA LCMS HNMR

Halopemide

Catalog No. T15461Cas No. 59831-65-1

Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.

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Pack Size	Price	Availability
1 mg	$50	In Stock
5 mg	$128	In Stock
10 mg	$213	In Stock
25 mg	$428	In Stock
50 mg	$639	In Stock
100 mg	$890	In Stock
1 mL x 10 mM (in DMSO)	$143	In Stock

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Product Introduction

Bioactivity

Description	Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.
Targets&IC50	PLD1:220 nM, PLD2:310 nM
In vitro	In transdifferentiated MOVAS cells, Halopemide (1-2 μM; 21 days) influences calcification[1].
In vivo	In the majority of monkeys tested, Halopemide (10 mg/kg; p.o.) causes dyskinesias[2].

Chemical Properties

Molecular Weight	416.88
Formula	C21H22ClFN4O2
Cas No.	59831-65-1

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 55 mg/mL (131.93 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.3988 mL	11.9939 mL	23.9877 mL	119.9386 mL
5 mM	0.4798 mL	2.3988 mL	4.7975 mL	23.9877 mL
10 mM	0.2399 mL	1.1994 mL	2.3988 mL	11.9939 mL
20 mM	0.1199 mL	0.5997 mL	1.1994 mL	5.9969 mL
50 mM	0.0480 mL	0.2399 mL	0.4798 mL	2.3988 mL
100 mM	0.0240 mL	0.1199 mL	0.2399 mL	1.1994 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc