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BMS-641988
BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
Catalog No. T67818Cas No. 1093276-09-5
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Purity:100%
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BMS-641988
Catalog No. T67818Cas No. 1093276-09-5
BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $163 | In Stock | |
| 5 mg | $400 | In Stock | |
| 10 mg | $600 | In Stock | |
| 25 mg | $959 | In Stock | |
| 50 mg | $1,280 | In Stock | |
| 100 mg | $1,750 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
| Description | BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer. |
| In vivo | Sixty-one men with CRPC were treated with daily BMS-641988 (5 to 150 mg). Seventeen of 23 evaluable patients (74%) exhibited stable disease on imaging (median 15 weeks; range 8-32), and 10 of 61 patients (16%) achieved a ≥ 30% decline in levels of prostate-specific antigen (PSA).[1] |
| Molecular Weight | 471.45 |
| Formula | C20H20F3N3O5S |
| Cas No. | 1093276-09-5 |
Storage & Solubility Information
| Storage | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 45 mg/mL (95.45 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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