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CB2R/FAAH modulator-3

CB2R/FAAH modulator-3 (compound 27) is a modulator targeting CB2R and FAAH, acting as a CB2R agonist with a Ki value of 20.1 nM and a CB1R agonist with a Ki value of 67.6 nM, while inhibiting FAAH with an IC50 value of 3.4 μM. This compound has research value in cancer, neurodegenerative disease-related inflammatory cascades, and COVID-19 infection.

Catalog No. T67747Cas No. 2876918-67-9

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Purity:99.02%

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COA HPLC HNMR

CB2R/FAAH modulator-3

Catalog No. T67747Cas No. 2876918-67-9

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Pack Size	Price	Availability
1 mg	$38	In Stock
5 mg	$89	In Stock
10 mg	$139	In Stock
25 mg	$278	In Stock
50 mg	$455	In Stock
100 mg	$672	In Stock
500 mg	$1,430	In Stock
1 mL x 10 mM (in DMSO)	$97	In Stock

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Product Introduction

Bioactivity

Description	CB2R/FAAH modulator-3 (compound 27) is a modulator targeting CB2R and FAAH, acting as a CB2R agonist with a Ki value of 20.1 nM and a CB1R agonist with a Ki value of 67.6 nM, while inhibiting FAAH with an IC50 value of 3.4 μM. This compound has research value in cancer, neurodegenerative disease-related inflammatory cascades, and COVID-19 infection.
In vitro	CB2R/FAAH modulator-3 (compound 27) at 10 μM reduces production of the inflammatory cytokines TNFα, IFN-γ, IL-1β, and IL-6 in unstimulated monocytes and macrophages[1].

Chemical Properties

Molecular Weight	341.49
Formula	C₂₂H₃₁NO₂
Cas No.	2876918-67-9

Storage & Solubility Information

Storage

Shipping with blue ice.

Solubility Information

DMSO: 50 mg/mL (146.42 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9283 mL	14.6417 mL	29.2834 mL	146.4172 mL
5 mM	0.5857 mL	2.9283 mL	5.8567 mL	29.2834 mL
10 mM	0.2928 mL	1.4642 mL	2.9283 mL	14.6417 mL
20 mM	0.1464 mL	0.7321 mL	1.4642 mL	7.3209 mL
50 mM	0.0586 mL	0.2928 mL	0.5857 mL	2.9283 mL
100 mM	0.0293 mL	0.1464 mL	0.2928 mL	1.4642 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

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