Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 has research value related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 38.00 | |
5 mg | In stock | $ 89.00 | |
10 mg | In stock | $ 139.00 | |
25 mg | In stock | $ 278.00 | |
50 mg | In stock | $ 455.00 | |
100 mg | In stock | $ 672.00 | |
500 mg | In stock | $ 1,430.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 97.00 |
Description | CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 has research value related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection. |
In vitro | CB2R/FAAH modulator-3 (compound 27)(10 μM) can reduce the production of the inflammatory cytokine TNFα、 IFN-γ、 IL-1β and IL6 in unstimulated monocytes and macrophages[1]. |
Molecular Weight | 341.49 |
Formula | C22H31NO2 |
CAS No. | 2876918-67-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (146.42 mM)
You can also refer to dose conversion for different animals. More
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CB2R/FAAH modulator-3 2876918-67-9 GPCR/G Protein Metabolism Neuroscience Cannabinoid Receptor FAAH CB2R/FAAHmodulator3 inhibitor inhibit