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VPC-13566

🥰Excellent
Catalog No. T29111Cas No. 218464-59-6

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.

VPC-13566

VPC-13566

🥰Excellent
Purity: 99.37%
Catalog No. T29111Cas No. 218464-59-6
VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.
Pack SizePriceAvailabilityQuantity
1 mg$40In Stock
2 mg$59In Stock
5 mg$98In Stock
10 mg$163In Stock
25 mg$347In Stock
50 mg$569In Stock
100 mg$892In Stock
500 mg$1,820In Stock
1 mL x 10 mM (in DMSO)$116In Stock
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Purity:99.37%
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Product Introduction

Bioactivity
Description
VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.
Chemical Properties
Molecular Weight258.32
FormulaC18H14N2
Cas No.218464-59-6
SmilesCC1=C2C(C(=CN2)C3=NC4=C(C=C3)C=CC=C4)=CC=C1
Relative Density.1.225 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 65 mg/mL (251.63 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.8712 mL19.3558 mL38.7117 mL193.5584 mL
5 mM0.7742 mL3.8712 mL7.7423 mL38.7117 mL
10 mM0.3871 mL1.9356 mL3.8712 mL19.3558 mL
20 mM0.1936 mL0.9678 mL1.9356 mL9.6779 mL
50 mM0.0774 mL0.3871 mL0.7742 mL3.8712 mL
100 mM0.0387 mL0.1936 mL0.3871 mL1.9356 mL

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