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LY2452473
Catalog No. T15804Cas No. 1029692-15-6
Alias OPK-88004, OPK 88004, LY-2452473, LY 2452473
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.
LY2452473
Catalog No. T15804Alias OPK-88004, OPK 88004, LY-2452473, LY 2452473Cas No. 1029692-15-6
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $38 | In Stock | |
| 5 mg | $89 | In Stock | |
| 10 mg | $122 | In Stock | |
| 25 mg | $163 | In Stock | |
| 50 mg | $198 | In Stock | |
| 100 mg | $328 | In Stock | |
| 500 mg | $787 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $98 | In Stock |
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CitedSelect Batch
Purity:99.72%
Contact us for more batch information
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer. |
| In vivo | METHODS: The disposition and metabolism of LY2452473 in humans was characterized following a single oral dose of 15 mg (100 μCi) of [¹⁴C]LY2452473 in six healthy male subjects. RESULTS: LY2452473 was rapidly absorbed (time to maximum plasma concentrations of LY2452473 and total radioactivity was 2-3 hours) and slowly eliminated (plasma terminal half-life of 27 hours, duration of LY2452473 and total radioactivity of 51 hours). [1] |
| Alias | OPK-88004, OPK 88004, LY-2452473, LY 2452473 |
| Molecular Weight | 374.44 |
| Formula | C22H22N4O2 |
| Cas No. | 1029692-15-6 |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 60 mg/mL (160.24 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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