Shopping Cart

Remove All

Your shopping cart is currently empty

Ralaniten triacetate

Select Batch

Purity:99.37%

ee:97.98%

Resource Download

COA CSFC HNMR HPLC HRMS LCMS

Ralaniten triacetate

Catalog No. T36375Cas No. 1637573-04-6

Ralaniten triacetate (EPI-506), a precursor of Ralaniten, is a first-of-its-kind, orally active androgen receptor N-terminal structural domain (AR-NTD) inhibitor with anticancer activity and can be used to study prostate and breast cancer.

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Pack Size	Price	Availability
1 mg	$165	In Stock
5 mg	$413	In Stock
10 mg	$689	In Stock
25 mg	$1,490	In Stock
50 mg	$1,980	In Stock
100 mg	$2,500	In Stock
1 mL x 10 mM (in DMSO)	$473	In Stock

Bulk & Custom

Add to Cart

Questions

Product Introduction

Bioactivity

Description	Ralaniten triacetate (EPI-506), a precursor of Ralaniten, is a first-of-its-kind, orally active androgen receptor N-terminal structural domain (AR-NTD) inhibitor with anticancer activity and can be used to study prostate and breast cancer.
In vitro	Ralaniten triacetate (EPI-506) is a highly specific small molecule targeting the N-terminal domain (NTD) of the androgen receptor (AR). It is commonly used in research on metastatic castration-resistant prostate cancer (mCRPC), where resistance to androgen deprivation therapy has developed[2].
Alias	EPI-506

Chemical Properties

Molecular Weight	521.00
Formula	C27H33ClO8
Cas No.	1637573-04-6

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 80 mg/mL (153.55 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.9194 mL	9.5969 mL	19.1939 mL	95.9693 mL
5 mM	0.3839 mL	1.9194 mL	3.8388 mL	19.1939 mL
10 mM	0.1919 mL	0.9597 mL	1.9194 mL	9.5969 mL
20 mM	0.0960 mL	0.4798 mL	0.9597 mL	4.7985 mL
50 mM	0.0384 mL	0.1919 mL	0.3839 mL	1.9194 mL
100 mM	0.0192 mL	0.0960 mL	0.1919 mL	0.9597 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

You can also refer to dose conversion for different animals. More

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc