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CCTA-1523

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Catalog No. T9587Cas No. 1616271-41-0

CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.

CCTA-1523

CCTA-1523

🥰Excellent
Purity: 99.03%
Catalog No. T9587Cas No. 1616271-41-0
CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.
Pack SizePriceAvailabilityQuantity
1 mg84 €In Stock
5 mg191 €In Stock
10 mg283 €In Stock
25 mg452 €In Stock
50 mg644 €In Stock
100 mg866 €In Stock
200 mg1.130 €In Stock
1 mL x 10 mM (in DMSO)192 €In Stock
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Purity:99.03%
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Product Introduction

Bioactivity
Description
CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.
In vitro
CCTA-1523 (5μM) sensitized the ABCG2 overexpressing cancer cells and ABCG2 transfected cells to the substrate chemotherapeutic drugs[1].
In vivo
Co-administration of CCTA-1523 restored the in vivo antitumor activity of doxorubicin in ABCG2 overexpressing tumor xenografts[1].
Chemical Properties
Molecular Weight340.2
FormulaC16H15Cl2NO3
Cas No.1616271-41-0
SmilesO(C)C=1C=C(C=CC1OC)C2=CC(NC(C(Cl)Cl)=O)=CC=C2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 50 mg/mL (146.97 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.9394 mL14.6972 mL29.3945 mL146.9724 mL
5 mM0.5879 mL2.9394 mL5.8789 mL29.3945 mL
10 mM0.2939 mL1.4697 mL2.9394 mL14.6972 mL
20 mM0.1470 mL0.7349 mL1.4697 mL7.3486 mL
50 mM0.0588 mL0.2939 mL0.5879 mL2.9394 mL
100 mM0.0294 mL0.1470 mL0.2939 mL1.4697 mL

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