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Almorexant

🥰Excellent
Catalog No. T2613Cas No. 871224-64-5
Alias ACT 078573

Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.

Almorexant

Almorexant

🥰Excellent
Purity: 98.02%
Catalog No. T2613Alias ACT 078573Cas No. 871224-64-5
Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
Pack SizePriceAvailabilityQuantity
1 mg$39In Stock
5 mg$90In Stock
10 mg$146In Stock
25 mg$333In Stock
50 mg$549In Stock
100 mg$798In Stock
1 mL x 10 mM (in DMSO)$98In Stock
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Purity:98.02%
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Product Introduction

Bioactivity
Description
Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
Targets&IC50
OX1:1.3 nM(ki), OX2:0.17 nM(ki)
AliasACT 078573
Chemical Properties
Molecular Weight512.56
FormulaC29H31F3N2O3
Cas No.871224-64-5
SmilesC(CC1=CC=C(C(F)(F)F)C=C1)[C@H]2C=3C(=CC(OC)=C(OC)C3)CCN2[C@@H](C(NC)=O)C4=CC=CC=C4
Relative Density.1.205
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 45 mg/mL (87.79 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.9510 mL9.7550 mL19.5099 mL97.5496 mL
5 mM0.3902 mL1.9510 mL3.9020 mL19.5099 mL
10 mM0.1951 mL0.9755 mL1.9510 mL9.7550 mL
20 mM0.0975 mL0.4877 mL0.9755 mL4.8775 mL
50 mM0.0390 mL0.1951 mL0.3902 mL1.9510 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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