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CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT (IC50s: 16 nM, 32 nM) with potent in vitro cellular activity in a wide range of cancer cells.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $223 | Backorder | |
10 mg | $346 | Backorder | |
50 mg | $971 | Backorder | |
100 mg | $1,323 | Backorder | |
200 mg | Inquiry | Backorder | |
500 mg | Inquiry | Backorder | |
1 mL x 10 mM (in DMSO) | $295 | Backorder |
Description | CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT (IC50s: 16 nM, 32 nM) with potent in vitro cellular activity in a wide range of cancer cells. |
Targets&IC50 | DNMT3B:1000 nM, G9a:16 nM, DNMT3A:92 nM, DNA methyltransferase:32 nM, DNMT1:1.5 nM (kd) |
Alias | CM-579 trihydrochloride |
Molecular Weight | 602.04 |
Formula | C29H43Cl3N4O3 |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
Solubility Information | H2O: 37.5 mg/mL (62.29 mM), Sonication is recommended. DMSO: 125 mg/mL (207.63 mM), Sonication is recommended. MEthanol: 75 mg/mL (124.58 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||||||||||||
H2O/MEthanol/DMSO
MEthanol/DMSO
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