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CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT (IC50s: 16 nM, 32 nM) with potent in vitro cellular activity in a wide range of cancer cells.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,520 | 8-10 weeks | |
50 mg | $1,980 | 8-10 weeks | |
100 mg | $2,500 | 8-10 weeks |
Description | CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT (IC50s: 16 nM, 32 nM) with potent in vitro cellular activity in a wide range of cancer cells. |
Targets&IC50 | G9a:16 nM, DNMT3B:1000 nM, DNMT1:1.5 nM (kd), DNMT3A:92 nM, DNA methyltransferase:32 nM |
Alias | CM-579 trihydrochloride |
Molecular Weight | 602.04 |
Formula | C29H43Cl3N4O3 |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
Solubility Information | H2O: 37.5 mg/mL (62.29 mM), Sonication is recommended. DMSO: 125 mg/mL (207.63 mM), Sonication is recommended. MEthanol: 75 mg/mL (124.58 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||||||||||||
H2O/MEthanol/DMSO
MEthanol/DMSO
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