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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $34 | In Stock | |
5 mg | $80 | In Stock | |
10 mg | $128 | In Stock | |
25 mg | $289 | In Stock | |
50 mg | $455 | In Stock | |
100 mg | $690 | In Stock | |
500 mg | $1,450 | In Stock |
Description | BAY-0069 is a potent and selective PPARγ transactivator that inhibits human PPARγ and murine PPARγ with IC50s of 6.3 nM and 24 nM, respectively.BAY-0069 can be used in cancer research. |
In vitro | BAY-0069 (0.0001, 0.001, 0.01, 0.01 and 1 μM; 7 days) leads to antiproliferative effects in the PPARγ-amplified cell line UM-UC-9.[1] |
In vivo | BAY-0069 (1 μM; 1 h) shows excellent microsomal stability with CL(b,hmic) of 0.47 L/h/kg in human liver microsomes and CL(b,rhep) of 3.9 L/h/kg in rat liver hepatocytes.[1] |
Molecular Weight | 466.28 |
Formula | C22H16BrN3O4 |
Cas No. | 420826-65-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 90.0 mg/mL (193.0 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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