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S1PR1 modulator 1
🥰Excellent
Catalog No. T12821Cas No. 2328109-05-1
S1PR1 modulator 1 is a selective inhibitor of S1PR1, with a pIC50 of 7.6.
S1PR1 modulator 1
🥰Excellent
Purity: 99.44%
Catalog No. T12821Cas No. 2328109-05-1
S1PR1 modulator 1 is a selective inhibitor of S1PR1, with a pIC50 of 7.6.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $59 | In Stock | |
| 5 mg | $122 | In Stock | |
| 10 mg | $173 | In Stock | |
| 25 mg | $285 | In Stock | |
| 50 mg | $422 | In Stock | |
| 100 mg | $626 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $141 | In Stock |
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Purity:99.44%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | S1PR1 modulator 1 is a selective inhibitor of S1PR1, with a pIC50 of 7.6. |
| Targets&IC50 | S1PR3:6(pIC50), S1PR1:7.6(pIC50) |
| In vitro | S1PR1 modulator 1 shows >40- and >80-fold selectivity, over the other S1PR isoforms S1PR3 (pIC50, 6), S1PR2 and S1PR4 (pIC50s, <5)[1]. |
| Molecular Weight | 408.51 |
| Formula | C23H24N2O3S |
| Cas No. | 2328109-05-1 |
| Smiles | N(\CCC)=C\1/N(C(=O)\C(=C\C2=CC(C)=C(OC(C)=O)C=C2)\S1)C3=C(C)C=CC=C3 |
| Relative Density. | 1.18 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 6.11 mg/mL (14.96 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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