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Selodenoson
🥰Excellent
Catalog No. T28748Cas No. 110299-05-3
Alias RG-14202, RG14202, DTI-0009, DTI0009, DT-009, DT009
Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
Selodenoson
🥰Excellent
Purity: 99.33%
Catalog No. T28748Alias RG-14202, RG14202, DTI-0009, DTI0009, DT-009, DT009Cas No. 110299-05-3
Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 126 € | In Stock | |
| 5 mg | 304 € | In Stock | |
| 10 mg | 446 € | In Stock | |
| 25 mg | 733 € | In Stock | |
| 50 mg | 1.026 € | In Stock | |
| 100 mg | 1.387 € | In Stock | |
| 500 mg | 2.774 € | In Stock |
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Purity:99.33%
ee:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias. |
| In vivo | Selodenoson (2, 4, 6, 8, 10, and 12 μg/kg; i.v.) provided for effective ventricular rate control in a dose-dependent manner with minimal side effects.[1] |
| Alias | RG-14202, RG14202, DTI-0009, DTI0009, DT-009, DT009 |
| Molecular Weight | 376.41 |
| Formula | C17H24N6O4 |
| Cas No. | 110299-05-3 |
| Smiles | O[C@H]1[C@H](N2C=3C(N=C2)=C(NC4CCCC4)N=CN3)O[C@H](C(NCC)=O)[C@H]1O |
| Relative Density. | 1.68g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 50 mg/mL (132.83 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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