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STING-IN-3
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STING-IN-3
Catalog No. T9029Cas No. 2244881-69-2
STING-IN-3 (C-171) is an inhibitor of stimulator of interferon genes (STING). It binds to STING, inhibits its palmitoylation, and prevents the recruitment and phosphorylation of TBK1.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | $45 | In Stock | |
| 25 mg | $85 | In Stock | |
| 50 mg | $134 | In Stock | |
| 100 mg | $207 | In Stock | |
| 200 mg | $310 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $51 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | STING-IN-3 (C-171) is an inhibitor of stimulator of interferon genes (STING). It binds to STING, inhibits its palmitoylation, and prevents the recruitment and phosphorylation of TBK1. |
| In vitro | C-171 binds to STING, inhibits its palmitoylation, and prevents the recruitment and phosphorylation of TBK1. It selectively reduces human and mouse STING-, but not RIG-I or TBK1-, mediated IFN-β reporter activity in HEK293 cells when used at concentrations ranging from 0.02 to 2 μM[1]. |
| Alias | C-171 |
| Molecular Weight | 316.35 |
| Formula | C17H20N2O4 |
| Cas No. | 2244881-69-2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||
| Solubility Information | DMSO: 3.16 mg/mL (10 mM)  | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
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