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Sinitrodil
🥰Excellent
Catalog No. T34648Cas No. 143248-63-9
Alias ITF-296, ITF296, ITF 296
Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.
Sinitrodil
🥰Excellent
Purity: 99%
Catalog No. T34648Alias ITF-296, ITF296, ITF 296Cas No. 143248-63-9
Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 134 € | In Stock | |
| 5 mg | 332 € | In Stock | |
| 10 mg | 503 € | In Stock | |
| 25 mg | 816 € | In Stock | |
| 50 mg | 1.121 € | In Stock | |
| 100 mg | 1.510 € | In Stock | |
| 500 mg | 3.030 € | In Stock | |
| 1 mL x 10 mM (in DMSO) | 401 € | In Stock |
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Purity:99%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris. |
| In vivo | Sinitrodil (10、20、40 mg; oral) increased gradually brachial artery compliance with increasing doses of sinitrodil (by 10, 20, and 27% with 10, 20, and 40 mg sinitrodil, respectively). Total peripheral resistance index decreased with isosorbide dinitrate (by 11%) and 40 mg sinitrodil (by 7%), while it remained unchanged with 10 mg and 20 mg sinitrodil.[3] |
| Alias | ITF-296, ITF296, ITF 296 |
| Molecular Weight | 238.2 |
| Formula | C10H10N2O5 |
| Cas No. | 143248-63-9 |
| Smiles | O=C1C=2C(OCN1CCON(=O)=O)=CC=CC2 |
| Relative Density. | 1.388g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 27.5 mg/mL (58.27 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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