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Ziconotide Acetate (107452-89-1 free base)

Catalog No. TP1559L CAS 914454-03-8

Synonyms: Prialt, Ziconotide Acetate

Ziconotide Acetate (107452-89-1 free base) (Prialt) is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide Acetate (107452-89-1 free base) acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.

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Ziconotide Acetate (107452-89-1 free base) Chemical Structure

Ziconotide Acetate (107452-89-1 free base), CAS 914454-03-8

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1 mg	In stock	$ 175.00
5 mg	In stock	$ 372.00
10 mg	In stock	$ 538.00
25 mg	In stock	$ 857.00
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Purity: 99.52%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	Prialt, Ziconotide Acetate
Molecular Weight	2639.2
Formula	C102H172N36O32S7
CAS No.	914454-03-8

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Brinzeu A, Berthiller J, Caillet JB, Staquet H, Mertens P. Ziconotide for spinal cord injury-related pain. Eur J Pain. 2019;23(9):1688-1700. doi:10.1002/ejp.1445

Citations

1. Dong Y, Gao Y, Xu S, et al. Closed-state inactivation and pore-blocker modulation mechanisms of human CaV2. 2. Cell Reports. 2021, 37(5): 109931.

Related compound libraries

This product is contained In the following compound libraries：

Peptide Compound Library Cyclic Peptide Library Macrocyclic Compound Library Approved Drug Library

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Keywords

Ziconotide Acetate (107452-89-1 free base) 914454-03-8 Membrane transporter/Ion channel Metabolism Calcium Channel analgesic non-opioid Ziconotide Acetate (107452891 free base) transmission SNX111 Inhibitor calcium Ziconotide Acetate 107452-89-1 free base Ca channels Ca2+ channels Prialt synaptic Ziconotide Ziconotide Acetate intrathecal 107452-89-1 N-type SNX-111 SNX 111 channels inhibit Ziconotide Acetate (107452 89 1 free base) inhibitor

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