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BD1063 dhydrochloride

🥰Excellent
Catalog No. T7488Cas No. 206996-13-6
Alias BD1063 2HCL

BD1063 dihydrochloride is a potent and selective sigma 1 (σ1) receptor antagonist (Ki = 9 nM).

BD1063 dhydrochloride

BD1063 dhydrochloride

🥰Excellent
Purity: 99.52%
Catalog No. T7488Alias BD1063 2HCLCas No. 206996-13-6
BD1063 dihydrochloride is a potent and selective sigma 1 (σ1) receptor antagonist (Ki = 9 nM).
Pack SizePriceAvailabilityQuantity
2 mg$41In Stock
5 mg$66In Stock
10 mg$92In Stock
25 mg$197In Stock
50 mg$357In Stock
100 mg$525In Stock
200 mg$739In Stock
500 mg$1,130In Stock
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Purity:99.52%
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Product Introduction

Bioactivity
Description
BD1063 dihydrochloride is a potent and selective sigma 1 (σ1) receptor antagonist (Ki = 9 nM).
In vivo
BD 1063 dose-dependently reduced ethanol self-administration in sP rats (3.3–11 mg/kg) and withdrawn, dependent Wistar rats (4–11 mg/kg) at doses that did not modify mean ethanol self-administration in non-dependent Wistar controls[1]
Animal Research
Rats (controls, N=11;?dependent, N=9) were pretreated with BD-1063 (0, 4.4, 7 and 11 mg/kg of body weight, free base weights) using a within-subject Latin square design.?sP rats: Rats (N=9) were pretreated with BD-1063 (0, 3, 4.4, 7 and 11 mg/kg of body weight, free base basis) using a within-subject Latin square design[1].
AliasBD1063 2HCL
Chemical Properties
Molecular Weight346.12
FormulaC13H20Cl4N2
Cas No.206996-13-6
SmilesCl.Cl.CN1CCN(CCc2ccc(Cl)c(Cl)c2)CC1
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
H2O: 50 mg/mL (144.46 mM)
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM2.8892 mL14.4459 mL28.8917 mL144.4586 mL
5 mM0.5778 mL2.8892 mL5.7783 mL28.8917 mL
10 mM0.2889 mL1.4446 mL2.8892 mL14.4459 mL
20 mM0.1445 mL0.7223 mL1.4446 mL7.2229 mL
50 mM0.0578 mL0.2889 mL0.5778 mL2.8892 mL
100 mM0.0289 mL0.1445 mL0.2889 mL1.4446 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
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2 Enter the in vivo formulation:
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