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CCG-63802

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Catalog No. T14897Cas No. 620112-78-9

CCG-63802 is a reversible small-molecule inhibitor of regulator of G protein signaling (RGS) proteins. CCG-63802 inhibits the interaction between RGS4 and Galpha with an IC50 value of 1.4 μM.

CCG-63802

CCG-63802

🥰Excellent
Catalog No. T14897Cas No. 620112-78-9
CCG-63802 is a reversible small-molecule inhibitor of regulator of G protein signaling (RGS) proteins. CCG-63802 inhibits the interaction between RGS4 and Galpha with an IC50 value of 1.4 μM.
Pack SizePriceAvailabilityQuantity
2 mg$36In Stock
5 mg$57In Stock
10 mg$97In Stock
25 mg$189In Stock
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Product Introduction

Bioactivity
Description
CCG-63802 is a reversible inhibitor of the regulator of G-protein signaling (RGS) protein and has the greatest potency at RGS4.
Targets&IC50
RGS4:1.4 μM
In vitro
CCG-63802 inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo.
Chemical Properties
Molecular Weight450.51
FormulaC26H18N4O2S
Cas No.620112-78-9
SmilesCc1cccc(Oc2nc3c(C)cccn3c(=O)c2\C=C(/C#N)c2nc3ccccc3s2)c1
Relative Density.1.31g/cm3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 1.67 mg/mL (3.71 mM), Sonication and heating are recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.2197 mL11.0985 mL22.1971 mL110.9853 mL

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