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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $132 | In Stock | |
5 mg | $328 | In Stock | |
10 mg | $538 | In Stock | |
25 mg | $1,130 | In Stock | |
50 mg | $1,890 | In Stock | |
100 mg | $2,500 | In Stock | |
1 mL x 10 mM (in DMSO) | $363 | In Stock |
Description | CDK12-IN-3 is a selective and potent CDK12 inhibitor with anti-tumor activity, which can be used to study malignant tumors. |
Targets&IC50 | CDK12:491 nM |
In vitro | CDK12-IN-3 is a highly selective inhibitor of CDK12, capable of effectively inhibiting the phosphorylation of Ser2 sites on the CTD repeat domain of RNA Polymerase II, exerting growth inhibitory effects on OV90 cells, and demonstrating acute cytotoxicity against THP1 cells[1]. |
Molecular Weight | 470.52 |
Formula | C23H28F2N8O |
Cas No. | 2220184-50-7 |
Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 200 mg/mL (425.06 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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