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CP-409092

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Catalog No. T10869LCas No. 194098-25-4

CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.

CP-409092

CP-409092

😃Good
Catalog No. T10869LCas No. 194098-25-4
CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
Pack SizePriceAvailabilityQuantity
25 mg$1,8208-10 weeks
50 mg$2,3808-10 weeks
100 mg$3,1008-10 weeks
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Product Introduction

Bioactivity
Description
CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
In vivo
[14C]CP-409,092(P.O.; 100 mg/kg; ) treatment, the total recovery is 89.1%+ or -3.2% for male rats and 89.3%+ or -0.58% for female rats. The pharmacokinetics of CP-409,092 (P.O.; 4 and 15 mg/kg;single intravenous) treatment , are characterized by high clearance of 169+ or -18 mL/min/kg, a volume of distribution of 8.99+ or -1.46 L/kg, and an oral bioavailability of 2.9%+ or -3%.
Chemical Properties
Molecular Weight297.35
FormulaC17H19N3O2
Cas No.194098-25-4
Relative Density.1.283 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 41.67 mg/mL (140.14 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.3630 mL16.8152 mL33.6304 mL168.1520 mL
5 mM0.6726 mL3.3630 mL6.7261 mL33.6304 mL
10 mM0.3363 mL1.6815 mL3.3630 mL16.8152 mL
20 mM0.1682 mL0.8408 mL1.6815 mL8.4076 mL
50 mM0.0673 mL0.3363 mL0.6726 mL3.3630 mL
100 mM0.0336 mL0.1682 mL0.3363 mL1.6815 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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