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Dihydrexidine
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Catalog No. T13463LCas No. 123039-93-0
Alias DAR-0100
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.
Dihydrexidine
😃Good
Catalog No. T13463LAlias DAR-0100Cas No. 123039-93-0
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,970 | 8-10 weeks | |
| 50 mg | $2,580 | 8-10 weeks | |
| 100 mg | $3,400 | 8-10 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity. |
| Targets&IC50 | D1 receptor:10 nM, D1 receptor:660 nM |
| In vivo | Dihydrexidine shows poor oral bioavailability. It also has a relatively short half-life of 1 to 2 h [3]. Dihydrexidine hydrochloride (3 mg/kg; i.p.) yields dopamine D1 receptor agonist effects in vivo [4]. |
| Alias | DAR-0100 |
| Molecular Weight | 267.32 |
| Formula | C17H17NO2 |
| Cas No. | 123039-93-0 |
| Relative Density. | 1.267g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
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