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LpxH-IN-AZ1
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Purity:99.26%
LpxH-IN-AZ1
Catalog No. T11876Cas No. 901260-40-0
LpxH-IN-AZ1 is a potent inhibitor of the UDP-2,3-diacylglucosamine pyrophosphate hydrolase, LpxH, and sulfonylpiperazine compounds.LpxH-IN-AZ1 exhibits antimicrobial activity and inhibits Klebsiella pneumoniae with an IC50 of 0.36 μM.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $50 | In Stock | |
| 5 mg | $122 | In Stock | |
| 10 mg | $193 | In Stock | |
| 25 mg | $455 | In Stock | |
| 50 mg | $669 | In Stock | |
| 100 mg | $953 | In Stock | |
| 500 mg | $1,920 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | LpxH-IN-AZ1 is a potent inhibitor of the UDP-2,3-diacylglucosamine pyrophosphate hydrolase, LpxH, and sulfonylpiperazine compounds.LpxH-IN-AZ1 exhibits antimicrobial activity and inhibits Klebsiella pneumoniae with an IC50 of 0.36 μM. |
| Targets&IC50 | LpxH (E. coli):0.14 μM, LpxH (Klebsiella pneumoniae):0.36 μM |
| In vitro | LpxH-IN-AZ1 (1 μM) inhibits K. pneumoniae LpxH activity by 75% and E. coli LpxH activity by 83% when 100 μM UDPDAGn is present[1]. Additionally, it exhibits IC50 values of 0.36 μM for K. pneumoniae LpxH and 0.14 μM for E. coli LpxH[1]. |
| Molecular Weight | 453.48 |
| Formula | C21H22F3N3O3S |
| Cas No. | 901260-40-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 4.53 mg/mL (10 mM), Sonication is recommended.  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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