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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $34 | In Stock | |
2 mg | $48 | In Stock | |
5 mg | $80 | In Stock | |
10 mg | $113 | In Stock | |
25 mg | $233 | In Stock | |
50 mg | $449 | In Stock | |
100 mg | $659 | In Stock | |
500 mg | $1,390 | In Stock | |
1 mL x 10 mM (in DMSO) | $89 | In Stock |
Description | N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar potency to Enzalutamide and circulates at approximately the same plasma concentrations as enzalutamide. |
In vivo | N-desmethyl Enzalutamide is an active metabolite that is thought to contribute to the clinical effects of Enzalutamide Enzalutamide and circulates at approximately the same plasma concentrations as Enzalutamide.?The carboxylic acid metabolite is pharmacologically inactive and circulates at approximately 25 % lower plasma concentrations than Enzalutamide[1]. |
Alias | N-desmethyl MDV 3100 |
Molecular Weight | 450.41 |
Formula | C20H14F4N4O2S |
Cas No. | 1242137-16-1 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 50 mg/mL (111.01 mM) ![]() | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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