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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $34 | In Stock | |
5 mg | $78 | In Stock | |
10 mg | $119 | In Stock | |
25 mg | $239 | In Stock | |
50 mg | $355 | In Stock | |
100 mg | $527 | In Stock |
Description | NaV1.2/1.6 channel blocker-1 is a potent inhibitor of NaV1.2 and NaV1.6 channels, exhibiting inhibitory effects on rNaV1.6 and hNaV1.2. This compound can be utilized in the study of generalized epilepsy and movement disorders. |
Targets&IC50 | rNaV1.6:9.8 μM, Nav1.2 (human):24.4 μM |
In vitro | NaV1.2/1.6 channel blocker(Compound 13)inhibits 48.5% and 34.0% of NaV1.6 and NaV1.2 sodium currents, respectively, in HEK 293 cells stably expressing rat NaV1.6 and human NaV1.2 isoforms at concentrations ranging from 1 to 100 μM [1]. |
Molecular Weight | 258.34 |
Formula | C14H14N2OS |
Cas No. | 1199944-04-1 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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