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Tolperisone hydrochloride
🥰Excellent
Catalog No. T0511Cas No. 3644-61-9
Alias Tolperisone HCl, Muscalm, Midocalm
Tolperisone hydrochloride (Muscalm), a centrally acting muscle relaxant, is used in the therapy of pathologically increased tone of the cross-striated muscle resulted by neurological diseases (damage of the encephalomyelitis, myelopathy, multiple sclerosis, pyramidal tract) and of spastic paralysis and other encephalopathies manifested with muscular dystonia.
Tolperisone hydrochloride
🥰Excellent
Purity: 99.9%
Catalog No. T0511Alias Tolperisone HCl, Muscalm, MidocalmCas No. 3644-61-9
Tolperisone hydrochloride (Muscalm), a centrally acting muscle relaxant, is used in the therapy of pathologically increased tone of the cross-striated muscle resulted by neurological diseases (damage of the encephalomyelitis, myelopathy, multiple sclerosis, pyramidal tract) and of spastic paralysis and other encephalopathies manifested with muscular dystonia.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $29 | In Stock | |
| 50 mg | $34 | In Stock | |
| 100 mg | $48 | In Stock | |
| 200 mg | $69 | In Stock | |
| 500 mg | $118 | In Stock | |
| 1 g | $175 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $29 | In Stock |
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Purity:99.9%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tolperisone hydrochloride (Muscalm), a centrally acting muscle relaxant, is used in the therapy of pathologically increased tone of the cross-striated muscle resulted by neurological diseases (damage of the encephalomyelitis, myelopathy, multiple sclerosis, pyramidal tract) and of spastic paralysis and other encephalopathies manifested with muscular dystonia. |
| In vivo | Tolperisone hydrochloride is a safe and effective drug for the treatment of pain-reflex muscle spasms without the typical side effects of central muscle relaxants.Tolperisone blocks calcium ion flow in snail neurons, decreases sodium-potassium ion permeability at frog Lang's ganglion, and has an current passage through Nav1.6 channels (heterologous expression) Inhibitory effect on current through Nav1.6 channel (heterologous expression). |
| Alias | Tolperisone HCl, Muscalm, Midocalm |
| Molecular Weight | 281.82 |
| Formula | C16H24ClNO |
| Cas No. | 3644-61-9 |
| Smiles | Cl.CC(CN1CCCCC1)C(=O)C1=CC=C(C)C=C1 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 55 mg/mL (195.16 mM)  Ethanol: 52 mg/mL (184.5 mM) H2O: 51 mg/mL (181 mM) | |||||||||||||||||||||||||||||||||||
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H2O/Ethanol/DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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