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P2X4 antagonist-1
🥰Excellent
Catalog No. T87086Cas No. 2055601-42-6
P2X4 antagonist-1 is a potent P2X4 receptor antagonist used in the study of neurological, cardiovascular, and immune system diseases.
P2X4 antagonist-1
🥰Excellent
Catalog No. T87086Cas No. 2055601-42-6
P2X4 antagonist-1 is a potent P2X4 receptor antagonist used in the study of neurological, cardiovascular, and immune system diseases.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $48 | In Stock | |
| 5 mg | $113 | In Stock | |
| 10 mg | $179 | In Stock | |
| 25 mg | $355 | In Stock | |
| 50 mg | $569 | In Stock | |
| 100 mg | $892 | In Stock | |
| 200 mg | $1,220 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | P2X4 antagonist-1 is a potent P2X4 receptor antagonist used in the study of neurological, cardiovascular, and immune system diseases. |
| Targets&IC50 | P2X4 receptor:15 nM |
| In vitro | P2X4 antagonist-1 (Compound 24) is an antagonist targeting the P2X4 receptor with an IC50 of 15 nM. [1] |
| Molecular Weight | 485.77 |
| Formula | C20H15Cl3N2O4S |
| Cas No. | 2055601-42-6 |
| Smiles | O=C(NC1=CC=C(OC=2C=CC=C(Cl)C2)C(=C1)S(=O)(=O)N)CC=3C(Cl)=CC=CC3Cl |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (164.69 mM), Sonication is recommended | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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