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VPC171
🥰Excellent
Catalog No. T29112Cas No. 1018830-99-3
Alias VPC-171, VPC 171
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
VPC171
🥰Excellent
Purity: 99.52%
Catalog No. T29112Alias VPC-171, VPC 171Cas No. 1018830-99-3
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $67 | In Stock | |
| 2 mg | $88 | In Stock | |
| 5 mg | $133 | In Stock | |
| 10 mg | $191 | In Stock | |
| 25 mg | $353 | In Stock | |
| 50 mg | $492 | In Stock | |
| 100 mg | $696 | In Stock | |
| 200 mg | $938 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $136 | In Stock |
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Purity:99.52%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM). |
| In vivo | VCP171 produced a greater inhibition of eEPSC amplitude of nerve-injury versus control animals in both lamina I and lamina II neurons[2]. |
| Alias | VPC-171, VPC 171 |
| Molecular Weight | 347.35 |
| Formula | C18H12F3NOS |
| Cas No. | 1018830-99-3 |
| Smiles | Nc1scc(c1C(=O)c1ccccc1)-c1cccc(c1)C(F)(F)F |
| Relative Density. | 1.345 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 55 mg/mL (158.34 mM), Sonication is recommended.  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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