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(R)-(-)-JQ1 Enantiomer

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Purity:98.03%

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COA HPLC HNMR

(R)-(-)-JQ1 Enantiomer

Catalog No. T19618Cas No. 1268524-71-5

(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1. (+)-JQ1 is a BET bromodomain inhibitor, acting on BRD4(1/2)(IC50 of 77 nM/33 nM in a cell-free assay)

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Pack Size	Price	Availability
1 mg	$32	In Stock
2 mg	$45	In Stock
5 mg	$73	In Stock
10 mg	$113	In Stock
25 mg	$197	In Stock
50 mg	$313	In Stock
100 mg	$513	In Stock
1 mL x 10 mM (in DMSO)	$80	In Stock

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Related Compound Libraries of "(R)-(-)-JQ1 Enantiomer"

Product Introduction

Bioactivity

Description

(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1. (+)-JQ1 is a BET bromodomain inhibitor, acting on BRD4(1/2)(IC50 of 77 nM/33 nM in a cell-free assay)

Chemical Properties

Molecular Weight	456.99
Formula	C23H25ClN4O2S
Cas No.	1268524-71-5

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 90 mg/mL (196.94 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1882 mL	10.9412 mL	21.8823 mL	109.4116 mL
5 mM	0.4376 mL	2.1882 mL	4.3765 mL	21.8823 mL
10 mM	0.2188 mL	1.0941 mL	2.1882 mL	10.9412 mL
20 mM	0.1094 mL	0.5471 mL	1.0941 mL	5.4706 mL
50 mM	0.0438 mL	0.2188 mL	0.4376 mL	2.1882 mL
100 mM	0.0219 mL	0.1094 mL	0.2188 mL	1.0941 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

You can also refer to dose conversion for different animals. More

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc