Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8 nM for MOP and 4.2 nM for NOP.BPR1M97 exhibits anti-injurious effects and antinociceptive effects.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 118.00 | |
5 mg | In stock | $ 296.00 | |
10 mg | In stock | $ 465.00 | |
25 mg | In stock | $ 837.00 | |
50 mg | In stock | $ 1,394.00 | |
100 mg | In stock | $ 1,880.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 227.00 |
Description | BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8 nM for MOP and 4.2 nM for NOP.BPR1M97 exhibits anti-injurious effects and antinociceptive effects. |
Targets&IC50 | NOP:4.2 nM (ki), MOP:1.8 nM (ki) |
In vivo | In a murine model of cancer pain, BPR1M97 (1.8 mg/kg; s.c.; once) demonstrates antinociception.[1] |
Molecular Weight | 349.25 |
Formula | C18H18Cl2N2O |
CAS No. | 2059904-66-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 225.0 mg/mL (644.2 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
BPR1M97 2059904-66-2 Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor BPR-1M97 inhibitor inhibit