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CAY 10465

Catalog No. T4607 CAS 688348-33-6

Synonyms: CAY10465, CAY10465 Exclusive

CAY 10465 is a selective and high-affinity AhR agonist, with a Ki of 0.2 nM, and shows no effect on estrogen receptor (Ki <100000 nM).

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CAY 10465, CAS 688348-33-6

Pack Size	Availability	Price/USD
1 mg	In stock	$ 30.00
2 mg	In stock	$ 44.00
5 mg	In stock	$ 70.00
10 mg	In stock	$ 112.00
25 mg	In stock	$ 239.00
50 mg	In stock	$ 453.00
100 mg	In stock	$ 687.00
1 mL * 10 mM (in DMSO)	In stock	$ 78.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description	CAY 10465 is a selective and high-affinity AhR agonist, with a Ki of 0.2 nM, and shows no effect on estrogen receptor (Ki >100000 nM).
Targets&IC50	ERR:>100000 nM(Ki), AhR:0.2 nM(Ki)

Synonyms	CAY10465, CAY10465 Exclusive
Molecular Weight	317.13
Formula	C15H9Cl2F3
CAS No.	688348-33-6

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 100 mg/mL (315.33 mM)

References and Literature

1. de Medina P, et al. Synthesis and biological properties of new stilbene derivatives of resveratrol as new selective aryl hydrocarbon modulators. J Med Chem. 2005 Jan 13;48(1):287-91. 2. Naem E, et al. Inhibition of apolipoprotein A-I gene by the aryl hydrocarbon receptor: a potential mechanism for smoking-associated hypoalphalipoproteinemia. Life Sci. 2012 Jul 26;91(1-2):64-9.

Related compound libraries

This product is contained In the following compound libraries：

Transcription Factor-Targeted Compound Library NO PAINS Compound Library Bioactive Compounds Library Max Bioactive Lipid Compound Library Bioactive Compound Library Nuclear Receptor Compound Library Anti-Metabolism Disease Compound Library Nonsteroidal Anti-Inflammatory Compound Library Immunology/Inflammation Compound Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

CAY 10465 688348-33-6 Immunology/Inflammation Metabolism Aryl Hydrocarbon Receptor AhR inhibit CAY-10465 Inhibitor CAY10465 CAY10465 Exclusive inhibitor

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.