Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selective and potent GPR142 antagonist.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 48.00 | |
5 mg | In stock | $ 116.00 | |
10 mg | In stock | $ 198.00 | |
25 mg | In stock | $ 349.00 | |
50 mg | In stock | $ 522.00 | |
100 mg | In stock | $ 743.00 | |
500 mg | In stock | $ 1,490.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 127.00 |
Description | CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selective and potent GPR142 antagonist. |
Targets&IC50 | BF3 (Androgen receptor):4 μM |
In vivo | I.p. administration of 30, 100 mg/kg CLP-3094 daily from Day 0 to Day 11 consistently displayed significantly lower severity of arthritis scores than vehicle-treated mice and reduced the arthritis scores dose-dependently, by not much.[2]. |
Synonyms | 2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE |
Molecular Weight | 304.79 |
Formula | C15H13ClN2OS |
CAS No. | 312749-73-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (328.09 mM)
You can also refer to dose conversion for different animals. More
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CLP-3094 312749-73-8 Endocrinology/Hormones Androgen Receptor LNCaP CLP3094 Inhibitor CLP 3094 inhibit 2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE prostate resistance antiandrogens cancer inhibitor