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CLP-3094

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Purity:99.84%

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COA HPLC HNMR

CLP-3094

Catalog No. T9179Cas No. 312749-73-8

CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selective and potent GPR142 antagonist.

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Pack Size	Price	Availability
1 mg	$48	In Stock
5 mg	$116	In Stock
10 mg	$198	In Stock
25 mg	$349	In Stock
50 mg	$522	In Stock
100 mg	$743	In Stock
500 mg	$1,490	In Stock
1 mL x 10 mM (in DMSO)	$127	In Stock

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Product Introduction

Bioactivity

Description	CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selective and potent GPR142 antagonist.
In vivo	I.p. administration of 30, 100 mg/kg CLP-3094 daily from Day 0 to Day 11 consistently displayed significantly lower severity of arthritis scores than vehicle-treated mice and reduced the arthritis scores dose-dependently, by not much.[2].
Alias	2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE

Chemical Properties

Molecular Weight	304.79
Formula	C15H13ClN2OS
Cas No.	312749-73-8

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 100 mg/mL (328.09 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.2809 mL	16.4047 mL	32.8095 mL	164.0474 mL
5 mM	0.6562 mL	3.2809 mL	6.5619 mL	32.8095 mL
10 mM	0.3281 mL	1.6405 mL	3.2809 mL	16.4047 mL
20 mM	0.1640 mL	0.8202 mL	1.6405 mL	8.2024 mL
50 mM	0.0656 mL	0.3281 mL	0.6562 mL	3.2809 mL
100 mM	0.0328 mL	0.1640 mL	0.3281 mL	1.6405 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

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