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Cyclosomatostatin Acetate
🥰Excellent
Catalog No. T21567L
Alias Cyclosomatostatin Acetate （84211-54-1 Free base）
Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell proliferation, ALDH+ cell population size, and sphere-formation in colorectal cancer cells.
Cyclosomatostatin Acetate
🥰Excellent
Purity: 98.83%
Catalog No. T21567LAlias Cyclosomatostatin Acetate （84211-54-1 Free base）
Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell proliferation, ALDH+ cell population size, and sphere-formation in colorectal cancer cells.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $153 | In Stock | |
| 2 mg | $265 | In Stock | |
| 5 mg | $392 | In Stock | |
| 10 mg | $598 | In Stock | |
| 25 mg | $888 | In Stock | |
| 50 mg | $1,190 | In Stock | |
| 100 mg | $1,610 | In Stock | |
| 200 mg | $2,170 | In Stock |
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Purity:98.83%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell proliferation, ALDH+ cell population size, and sphere-formation in colorectal cancer cells. |
| Alias | Cyclosomatostatin Acetate （84211-54-1 Free base） |
| Molecular Weight | 840.02 |
| Formula | C46H61N7O8 |
| Smiles | C[C@@H](OCC1=CC=CC=C1)[C@H]2C(NCCCCCCC(N[C@@H](CC3=CC=CC=C3)C(N[C@H](CC4=CNC5=CC=CC=C54)C(N[C@@H](CCCCN)C(N2)=O)=O)=O)=O)=O.CC(O)=O |
| Relative Density. | 1.31g/cm3 |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 8.4 mg/mL (10 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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