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Desmethyl cariprazine

Desmethyl cariprazine
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).
Catalog No. T15100Cas No. 839712-15-1

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Desmethyl cariprazine

Catalog No. T15100Cas No. 839712-15-1

Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).
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Product Introduction

Bioactivity
Description
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).
Targets&IC50
D3 receptor:0.085 nM (ki), D2 receptor:0.49 nM (ki), 5-HT1A receptor:2.6 nM (ki)
Chemical Properties
Molecular Weight413.38
FormulaC20H30Cl2N4O
Cas No.839712-15-1
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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