Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75). Glibornuride inhibits high affinity [3H]-glibenclamide binding with the potencies expected from their K+ channel activity.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 77.00 | |
2 mg | In stock | $ 113.00 | |
5 mg | In stock | $ 189.00 | |
10 mg | In stock | $ 297.00 | |
25 mg | In stock | $ 490.00 | |
50 mg | In stock | $ 728.00 | |
100 mg | In stock | $ 987.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 198.00 |
Description | Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75). Glibornuride inhibits high affinity [3H]-glibenclamide binding with the potencies expected from their K+ channel activity. |
Targets&IC50 | K+-ATP channel:5.75 (pKi) |
In vivo | Administration of Glibornuride (5 mg/kg; gavage, daily for 28 days) results in an enhance in body weights in the diabetic groups in Swiss albino rats. Administration of Glibornuride for 28 days, obviously enhances the liver lipid peroxidation levels in diabetic rats. Treatment with Glibornuride (28 days) reduces serum uric acid levels in diabetic rats [2]. |
Molecular Weight | 366.48 |
Formula | C18H26N2O4S |
CAS No. | 26944-48-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (682.17 mM)
You can also refer to dose conversion for different animals. More
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Glibornuride 26944-48-9 Membrane transporter/Ion channel Potassium Channel Inhibitor K channel KcsA blocker ATP sensitive inhibit Parsley Streptozotocin Antidiabetic inhibitor