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Nafarelin acetate(76932-56-4 free base)

Catalog No. T21309 CAS 76932-60-0

Synonyms: RS-94991-298, Nafarelin acetate, Nafarelin acetate hydrate, Synarel

Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH). It may be used in the treatment of estrogen-dependent conditions.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Nafarelin acetate(76932-56-4 free base) Chemical Structure

Nafarelin acetate(76932-56-4 free base), CAS 76932-60-0

Pack Size	Availability	Price/USD
5 mg	In stock	$ 50.00
10 mg	In stock	$ 75.00
25 mg	In stock	$ 128.00
50 mg	In stock	$ 192.00
100 mg	In stock	$ 287.00
200 mg	In stock	$ 431.00

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Purity: 99.98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	RS-94991-298, Nafarelin acetate, Nafarelin acetate hydrate, Synarel
Molecular Weight	1400.56
Formula	C68H89N17O16
CAS No.	76932-60-0

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: Insoluble

DMSO: Soluble

References and Literature

1. Ludwig C, Desmoulins PO, Driancourt MA, Goericke-Pesch S, Hoffmann B. Reversible downregulation of endocrine and germinative testicular function (hormonal castration) in the dog with the GnRH-agonist azagly-nafarelin as a removable implant "Gonazon"; a preclinical trial. Theriogenology. 2009 Apr 15;71(7):1037-45. 2. Cheng MH, Yu BK, Chang SP, Wang PH. A randomized, parallel, comparative study of the efficacy and safety of nafarelin versus danazol in the treatment of endometriosis in Taiwan. J Chin Med Assoc. 2005 Jul;68(7):307-14. PubMed PMID: 16038370. 3. Raiman J, Koljonen M, Huikko K, Kostiainen R, Hirvonen J. Delivery and stability of LHRH and Nafarelin in human skin: the effect of constant/pulsed iontophoresis. Eur J Pharm Sci. 2004 Feb;21(2-3):371-7. PubMed PMID: 14757511. 4. Suh J, Lee E, Hwang S, Yoon S, Yoon BK, Bae D, Choi D. Dose of GnRH agonist (nafarelin acetate) affects intrafollicular PAPP-A expression in controlled ovarian hyperstimulation cycle. Eur J Obstet Gynecol Reprod Biol. 2004 Jan 15;112(1):65-8. PubMed PMID: 14687742.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Approved Drug Library Anti-Cancer Drug Library Anti-Cancer Clinical Compound Library Peptide Compound Library NO PAINS Compound Library

Related Products

Related compounds with same targets

(R)-Elagolix Cetrorelix diacetate Lecirelin acetate(61012-19-9 free base) Ganirelix Acetate LGnRH-III, lamprey acetate(147859-97-0 free base) Alarelin Acetate Relugolix Histrelin acetate

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Nafarelin acetate(76932-56-4 free base) 76932-60-0 GPCR/G Protein GNRH Receptor RS-94991-298 Nafarelin acetate(76932564 free base) Nafarelin acetate Hydrate Nafarelin acetate(76932 56 4 free base) Nafarelin acetate Nafarelin acetate hydrate Nafarelin Acetate Synarel inhibitor inhibit

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