store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 700.00 | |
5 mg | In stock | $ 1,800.00 |
Description | Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity. |
Targets&IC50 | PRP:81 nM |
In vitro | In vitro, Nexopamil most potently inhibits serotonin-induced platelet aggregation in dog platelet-rich plasma (PRP) with an IC50 of 81 nM [1]. |
In vivo | Within the first 30 minutes after application, Nexopamil (0.05 mg/kg) completely abolishes cyclic flow reductions (CFRs) without significantly altering hemodynamics [1]. |
Synonyms | (Rac)-Nexopamil |
Molecular Weight | 404.59 |
Formula | C24H40N2O3 |
CAS No. | 116759-35-4 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Nexopamil racemate 116759-35-4 GPCR/G Protein Membrane transporter/Ion channel Metabolism Neuroscience 5-HT Receptor Calcium Channel (Rac)-Nexopamil inhibitor inhibit