Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,220.00 | |
50 mg | 6-8 weeks | $ 1,590.00 | |
100 mg | 6-8 weeks | $ 2,430.00 |
Description | Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM). |
In vivo | The metabolic pathway of Odapipam in phenobarbital-induced rat liver microsomes has been examined, revealing the formation of five distinct metabolites during its incubation. Analysis of the electron-ionization (EI+) mass spectra identified these metabolites as N-desmethyl-Odapipam, 1-hydroxy-Odapipam, two isomers of 3′-hydroxy-Odapipam, and a dehydrogenated metabolite within the dihydrobenzofuran moiety[1]. |
Synonyms | NNC 756 |
Molecular Weight | 329.82 |
Formula | C19H20ClNO2 |
CAS No. | 131796-63-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Odapipam 131796-63-9 GPCR/G Protein Neuroscience Dopamine Receptor NNC756 NNC 756 NNC-756 inhibitor inhibit