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PKR-IN-2

Catalog No. T12499 CAS 1628428-01-2

PKR-IN-2 is a activator of pyruvate kinase (PKR).

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PKR-IN-2, CAS 1628428-01-2

Pack Size	Availability	Price/USD
1 mg	In stock	$ 153.00
5 mg	In stock	$ 308.00
10 mg	In stock	$ 442.00
25 mg	In stock	$ 729.00
50 mg	In stock	$ 987.00
100 mg	In stock	$ 1,390.00
1 mL * 10 mM (in DMSO)	In stock	$ 323.00

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Purity: 99.17%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

PKR-IN-2 is a activator of pyruvate kinase (PKR).

Molecular Weight	468.57
Formula	C24H28N4O4S
CAS No.	1628428-01-2

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 45 mg/mL (96.04 mM), Sonification is recommended.

References and Literature

1. Popovici-Muller, et al. Preparation of N-(piperidinecarbonylphenyl) sulfonamide compounds as pyruvate kinase modulators. From PCT Int. Appl. (2014), WO2014139144A1 20140918. 2. Cianchetta Giovanni, et al. Preparation of aroylpiperidines, particularly arysulfonylamino and heteroarylsulfonylamino substituted, as pyruvate kinase PKM2 modulators useful in the treatment of cancer and compositions containing them. From PCT Int. Appl.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Active Compound Library Cuproptosis Compound Library Bioactive Compounds Library Max NO PAINS Compound Library Bioactive Compound Library Metabolism Compound Library Glutamine Metabolism Compound Library Kinase Inhibitor Library Glycometabolism Compound Library Anti-Cancer Metabolism Compound Library

Related Products

Related compounds with same targets

PKM2 activator 2 Mitapivat Dimethylaminomicheliolide HCl DL-Serine Shikonin Disodium monofluorophosphate DASA-58 PKM2 inhibitor G

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

PKR-IN-2 1628428-01-2 Metabolism PKM pyruvate PKRIN2 Pyruvate Kinase kinase PKR IN 2 inhibit Inhibitor deficiency inhibitor

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.