Search Result

Search Results for " kinase "

Targets

RIP kinase Aurora Kinase Haspin Kinase LIM Kinase Serine/threonin kinase S6 Kinase Glucokinase Casein Kinase Hexokinase AAK1 (AP2 associated kinase 1) Stemness kinase ROS Kinase Tyrosine Kinases Fer/FerT kinase Tie-2

3070

Compounds

251

Natural Products

1274

Recombinant Proteins

Libraries

Cat No.	Product Name	Synonyms	Targets
T6335	Tie2 kinase inhibitor 1	Tie2 kinase inhibitor	Tie-2
	Tie2 kinase inhibitor 1 (Tie2 kinase inhibitor), an optimized compound of SB-203580, is selective to Tie2 with IC50 of 0.25 μM, which is 200-fold more effective than p38.		Tie-2
T5524	Aurora kinase inhibitor-3	Aurora Kinase Inhibitor III	Aurora Kinase
	Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK, IGF-1R, c-Src, TRKB, SYK, and EGFR.		Aurora Kinase
T4191	Multi-kinase inhibitor 1	Multi-kinase inhibitor I	Others , Bcr-Abl , PDGFR , c-Kit
	Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.		Others , Bcr-Abl , PDGFR , c-Kit
T9040	Aurora kinase inhibitor-2	IUN-70219,Aurora Kinase Inhibitor II	Aurora Kinase
	Aurora kinase inhibitor-2 (IUN-70219) is a cell-permeable anilinoquinazoline that inhibit the activity of Aurora A (IC50 = 0.39 M).		Aurora Kinase
T10276L	AKT Kinase Inhibitor HCl	AKT Kinase Inhibitor HCl(842148-40-7 Free base)	Akt
	AKT Kinase Inhibitor HCl is an Akt inhibitor with antitumor activity.		Akt
T11184	EML4-ALK kinase inhibitor 1	EML4 ALK kinase inhibitor 1,EML4-ALK kinase inhibitor 1	ALK
	EML4-ALK kinase inhibitor 1 (EML4 ALK kinase inhibitor 1) is a potent oral active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (EML4-ALK), with an IC50 of 1 nM.		ALK
T60108	PDGFR Tyrosine Kinase Inhibitor III	PDGF Receptor Tyrosine Kinase Inhibitor III	PDGFR
	PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III) (PDGF Receptor Tyrosine Kinase Inhibitor III) is a multikinase inhibitor that inhibits PDGFR, EGFR, FGFR, PKA, and PKC, respectively. PDGF...		PDGFR
T16987	TAO Kinase inhibitor 1		Others , MAPK
	TAO Kinase inhibitor 1 delays mitosis and induces mitotic cell death. TAO Kinase inhibitor 1 is a selective and ATP-competitive thousand-and-one amino acid kinases inhibitor (IC50s: 11 to 15 nM for TAOK1 and 2, respectiv...		Others , MAPK
T8864	Thymidylate Kinase Inhibitor, YMU1		Others
	YMU1 is a human thymidylate kinase (hTMPK) inhibitor. YMU1 stabilizes the conformation of ligand-induced degradation (LID) region of hTMPK and blocks the catalytic site or ATP-binding site.		Others
TP1053L	Protein Kinase C 19-31 acetate	Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate	PKC
	Protein Kinase C 19-31 acetate, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is...		PKC
T12728	RIP2 Kinase Inhibitor 3		Others , RIP kinase
	RIP2 Kinase Inhibitor 3 is a potent and selective inhibitor of RIP2 with an IC50 of 1 nM.		Others , RIP kinase
T12721	Rho-Kinase-IN-1		ROCK
	Rho-Kinase-IN-1 is an inhibitor of ROCK with Kis of 30.5 nM and 3.9 nM for ROCK1 and ROCK2, respectively. Rho-Kinase-IN-1 can be used in studies about excessive cell proliferation, remodeling, edema and inflammation dise...		ROCK
T4692	Protein kinase inhibitors 1 hydrochlorid	Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))	Others
	Protein kinase inhibitors 1 hydrochlorid (Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))) is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.		Others
T9564	IRE1α kinase-IN-1		IRE1
	IRE1α kinase-IN-1 is a highly selective IRE1α (ERN1) inhibitor, with an IC50 of 77 nM. It displays 100-fold selectivity for IRE1α over the IRE1β isoform. It inhibits ER stress-induced IRE1α oligomerization and autophosph...		IRE1
T10276	AKT Kinase Inhibitor		Akt
	AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.		Akt
T10687	Casein Kinase II Inhibitor IV		Casein Kinase
	Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.		Casein Kinase
T64350	Casein kinase 1δ-IN-3		Casein Kinase
	Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) is a casein kinase 1 delta (CK1d) inhibitor with a pIC50 of 6.5376 M.		Casein Kinase
TP1051L	Protein Kinase C Peptide Substrate acetate	Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)	Others
	Protein Kinase C Peptide Substrate acetate targets specific cell spacers ina manner that is dependent on second messengers and specific adaptor proteins in response to extracellular signals that activate g protein-couple...		Others
T6409	ALK kinase inhibitor-1	SAR348830	Others
	SAR348830 is an ALK inhibitor, targeting anaplastic lymphoma kinase.		Others
T77500	Casein kinase 1δ-IN-6		Casein Kinase
	Casein kinase 1δ-IN-6 is a potent and selective inhibitor of the protein kinase CK-1δ with an IC50 of 23 nM.Casein kinase 1δ-IN-6 shows neuroprotective and anti-inflammatory activity in both in vitro and in vivo assays.C...		Casein Kinase
T64376	Casein kinase 1δ-IN-9		NADPH
	Casein kinase 1δ-IN-9 is a Quinone reductase 2 inhibitor with IC50 of 0.6μM.		NADPH
T67755	Protein kinase G inhibitor-1		PKA
	Protein kinase G inhibitor-1 is a potent Protein kinase G inhibitor, IC50= 0.9 uM.		PKA
T5466	Tyrosine kinase-IN-1		VEGFR , FGFR , FLT , PDGFR
	Tyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor（KDR, Flt-1, FGFR1 and PDGFRα with IC50s of 4nM, 20nM, 4nM, 2 nM ,respectively）		VEGFR , FGFR , FLT , PDGFR
T9175	Casein Kinase inhibitor A51		Apoptosis , Casein Kinase
	Casein Kinase inhibitor A51 is an orally active casein kinase 1α (CK1α) inhibitor with anticancer activity that induces apoptosis in leukemia cells, and may be used in the study of neck cancers, acute myeloid leukemia, b...		Apoptosis , Casein Kinase
T9631	IRAK-4 protein kinase inhibitor 2		IRAK
	IRAK-4 protein kinase inhibitor 2 is a potent interleukin-1 receptor-associated kinase-4 (IRAK-4) inhibitor(IC50 = 4 μM).		IRAK
TP1271L	Calmodulin-Dependent Protein Kinase II 290-309 acetate	Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)	CaMK
	Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).		CaMK
T9779	Protein kinase inhibitor 6
	Protein kinase inhibitor 6 is a protein kinase inhibitor.
T9940	Protein kinase G inhibitor-2		Others
	Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities.		Others
T77501	TAO Kinase inhibitor 2		Serine/threonin kinase
	TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.		Serine/threonin kinase
T60295	Casein kinase 1δ-IN-1	WAY-643895	Casein Kinase
	Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ. Casein kinase 1δ-IN-1 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.		Casein Kinase
TP1216	CaM kinase II inhibitor TFA salt	Autocamtide-2-related inhibitory peptide (TFA)	CaMK
	CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.		CaMK
T9229	Pim-1/2 kinase inhibitor 1		Pim
	Pim-1/2 Kinase Inhibitor 1, an orally active inhibitor, impedes the action of Pim kinases by preventing their ability to phosphorylate peptides. It particularly inhibits the phosphorylation of 4E-BP1 and p27 Kip1 by Pim ...		Pim
T77648	Casein kinase 1δ-IN-14	WAY-637081	Others
	Casein kinase 1δ-IN-14 (WAY-637081) can be used to study atherosclerosis-related cardiovascular disease.		Others
T77746	Tyrosine kinase-IN-7		EGFR , Antiviral
	Tyrosine kinase-IN-7 is a potent inhibitor of the tyrosine kinase EGFR, inhibiting EGFR(WT) and EGFR(T790M) and showing anti-cancer and anti-tumor activity in a variety of cancer cell lines. Tyrosine kinase-IN-7 has pote...		EGFR , Antiviral
T4026	SU5408	VEGFR2 Kinase Inhibitor I	VEGFR
	SU5408 (VEGFR2 Kinase Inhibitor I) is a potent, cell-permeable inhibitor of the VEGFR2 kinase.		VEGFR
T77708	Casein kinase 1δ-IN-7		Casein Kinase
	Casein kinase 1δ-IN-7 is a Casein kinase 1δ inhibitor for neurodegenerative diseases such as Alzheimer's disease.		Casein Kinase
T83627	Pim-1 kinase inhibitor 8		Pim , PKC
	Pim-1 kinase inhibitor 8 is a potent Pim-1 kinase inhibitor with anticancer activity and can effectively inhibit cell migration.Pim-1 kinase inhibitor 8 is cytotoxic to MCF-7 and HepG2 cells, and is a candidate compound ...		Pim , PKC
T60109	Protein kinase inhibitor H-7	5-(2-methylpiperazine-1-sulfonyl)isoquinoline,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine	PKC
	Protein kinase inhibitor H-7 (5-(2-methylpiperazine-1-sulfonyl)isoquinoline) is a potent inhibitor of protein kinase C (PKC) with a Ki of 6 μM. Protein kinase inhibitor H-7 is also a cyclic nucleotide dependent protein k...		PKC
T77709	Casein kinase 1δ-IN-8		Casein Kinase
	Casein kinase 1δ-IN-8 is an inhibitor of casein kinase 1δ and is used to treat neurodegenerative diseases such as Alzheimer's disease type.		Casein Kinase
T67944	P38 MAP Kinase Inhibitor Ⅵ		p38 MAPK
	p38 MAP Kinase Inhibitor Ⅵ is a potent p38 MAP Kinase inhibitor with anti-inflammatory activity.		p38 MAPK
T82174	HRIO2 kinase ligand-1		Others
	hRIO2 kinase ligand-1 is a potent ligand for hRIO2 kinase (Kd: 520 nM).		Others
T38841	IRE1α kinase-IN-2	IRE1α kinase-IN-2
	IRE1α kinase-IN-2 is a highly potent inhibitor of IRE1α kinase, demonstrating an EC50 of 0.82 μM. It effectively impedes IRE1α kinase autophosphorylation with an IC50 of 3.12 μM. Additionally, IRE1α kinase-IN-2 effective...
T40336	IRE1α kinase-IN-6	IRE1α kinase-IN-6
	IRE1α kinase-IN-6 is a potent IRE1α inhibitor with an IC 50 value of 4.4 nM.
T22831	Protein kinase inhibitor H-7 dihydrochloride	H-7 dihydrochloride	PKC
	Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor. Protein kinase inhibitor H-7 dihydrochloride (100 μM) significantly inhibits TPA (skin tumor promoter, 12-O-...		PKC
T39482	Casein Kinase inhibitor A86	Casein Kinase inhibitor A86
	Casein Kinase inhibitor A86 is a highly effective and orally bioavailable inhibitor of casein kinase 1α (CK1α). Additionally, it displays inhibitory actions towards CDK7 (TFIIH) and CDK9 (P-TEFb). Furthermore, Casein Kin...
T79860	TIE-2/VEGFR-2 kinase-IN-5		VEGFR , Tie-2
	TIE-2/VEGFR-2 kinase-IN-5 is a potent TIE-2 and VEGFR-2 tyrosine kinase receptor inhibitor with anti-angiogenic activity and is commonly used in biomedical research related to angiogenesis.		VEGFR , Tie-2
T35525	PI3-Kinase α Inhibitor 2	PI3-Kinase α Inhibitor 2
	Phosphatidylinositol 3-kinase (PI3K) catalyzes the phosphorylation of the 3' hydroxyl position of PIs to produce the second messengers PtdIns-(3,4)-P2 and PtdIns-(3,4,5)-P3. PI3Kα, β, and δ are class 1A enzymes composed ...
T77526	Pim-1 kinase inhibitor 4		Apoptosis , Pim
	Pim-1 kinase inhibitor 4 is a potent Pim-1 kinase inhibitor with an IC50 value of 17.01 nM.Pim-1 kinase inhibitor 4 also possesses antioxidant activity and potential anticancer activity, and inhibits DPPH.Pim-1 kinase in...		Apoptosis , Pim
T35526	PI3-Kinase α Inhibitor 2 (hydrochloride)	PI3-Kinase α Inhibitor 2 (hydrochloride)
	PI3-Kinase α Inhibitor 2 (hydrochloride) is a PI3-Kinase α inhibitor.
T37248	Pantothenate Kinase Inhibitor
	Pantothenate Kinase Inhibitor (PANKi) is a reversible inhibitor of pantothenate kinase (PanK; IC50s = 70, 92, and 25 nM for PanK1β, PanK2, and PanK3, respectively), the rate-limiting enzyme in the synthesis of coenzyme A...

Compounds

Tie2 kinase inhibitor 1

T6335

Synonym: Tie2 kinase inhibitor

Target: Tie-2

Aurora kinase inhibitor-3

T5524

Synonym: Aurora Kinase Inhibitor III

Target: Aurora Kinase

Multi-kinase inhibitor 1

T4191

Synonym: Multi-kinase inhibitor I

Target: Others, Bcr-Abl, PDGFR, c-Kit

Aurora kinase inhibitor-2

T9040

Synonym: IUN-70219,Aurora Kinase Inhibitor II

Target: Aurora Kinase

AKT Kinase Inhibitor HCl

T10276L

Synonym: AKT Kinase Inhibitor HCl(842148-40-7 Free base)

Target: Akt

EML4-ALK kinase inhibitor 1

T11184

Synonym: EML4 ALK kinase inhibitor 1,EML4-ALK kinase inhibitor 1

Target: ALK

PDGFR Tyrosine Kinase Inhibitor III

T60108

Synonym: PDGF Receptor Tyrosine Kinase Inhibitor III

Target: PDGFR

TAO Kinase inhibitor 1

T16987

Synonym:

Target: Others, MAPK

Thymidylate Kinase Inhibitor, YMU1

T8864

Synonym:

Target: Others

Protein Kinase C 19-31 acetate

TP1053L

Synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate

Target: PKC

RIP2 Kinase Inhibitor 3

T12728

Synonym:

Target: Others, RIP kinase

Protein kinase inhibitors 1 hydrochlorid

T4692

Synonym: Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))

AKT Kinase Inhibitor

T10276

Synonym:

Target: Akt

Casein Kinase II Inhibitor IV

T10687

Synonym:

Target: Casein Kinase

Casein kinase 1δ-IN-3

T64350

Synonym:

Target: Casein Kinase

Protein Kinase C Peptide Substrate acetate

TP1051L

Synonym: Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)

Target: Others

ALK kinase inhibitor-1

T6409

Synonym: SAR348830

Target: Others

Casein kinase 1δ-IN-6

T77500

Synonym:

Target: Casein Kinase

Casein kinase 1δ-IN-9

T64376

Synonym:

Target: NADPH

Protein kinase G inhibitor-1

T67755

Synonym:

Target: PKA

Tyrosine kinase-IN-1

T5466

Synonym:

Target: VEGFR, FGFR, FLT, PDGFR

Casein Kinase inhibitor A51

T9175

Synonym:

Target: Apoptosis, Casein Kinase

IRAK-4 protein kinase inhibitor 2

T9631

Synonym:

Target: IRAK

Calmodulin-Dependent Protein Kinase II 290-309 acetate

TP1271L

Synonym: Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)

Target: CaMK

Protein kinase inhibitor 6

T9779

Synonym:

Target:

Protein kinase G inhibitor-2

T9940

Synonym:

Target: Others

TAO Kinase inhibitor 2

T77501

Synonym:

Target: Serine/threonin kinase

Casein kinase 1δ-IN-1

T60295

Synonym: WAY-643895

Target: Casein Kinase

CaM kinase II inhibitor TFA salt

TP1216

Synonym: Autocamtide-2-related inhibitory peptide (TFA)

Target: CaMK

Pim-1/2 kinase inhibitor 1

T9229

Synonym:

Target: Pim

Casein kinase 1δ-IN-14

T77648

Synonym: WAY-637081

Target: Others

Tyrosine kinase-IN-7

T77746

Synonym:

Target: EGFR, Antiviral

SU5408

T4026

Synonym: VEGFR2 Kinase Inhibitor I

Target: VEGFR

Casein kinase 1δ-IN-7

T77708

Synonym:

Target: Casein Kinase

Pim-1 kinase inhibitor 8

T83627

Synonym:

Target: Pim, PKC

Protein kinase inhibitor H-7

T60109

Synonym: 5-(2-methylpiperazine-1-sulfonyl)isoquinoline,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine

Target: PKC

Casein kinase 1δ-IN-8

T77709

Synonym:

Target: Casein Kinase

p38 MAP Kinase Inhibitor Ⅵ

T67944

Synonym:

Target: p38 MAPK

hRIO2 kinase ligand-1

Synonym: IRE1α kinase-IN-2

Target:

IRE1α kinase-IN-6

T40336

Synonym: IRE1α kinase-IN-6

Target:

Protein kinase inhibitor H-7 dihydrochloride

T22831

Synonym: H-7 dihydrochloride

Target: PKC

Casein Kinase inhibitor A86

T39482

Synonym: Casein Kinase inhibitor A86

Target:

TIE-2/VEGFR-2 kinase-IN-5

T79860

Synonym:

Target: VEGFR, Tie-2

PI3-Kinase α Inhibitor 2

T35525

Synonym: PI3-Kinase α Inhibitor 2

Target:

Pim-1 kinase inhibitor 4

T77526

Synonym:

Target: Apoptosis, Pim

PI3-Kinase α Inhibitor 2 (hydrochloride)

T35526

Synonym: PI3-Kinase α Inhibitor 2 (hydrochloride)

Target:

Pantothenate Kinase Inhibitor

T37248

Synonym:

Target:

Cat No.	Product Name	Synonyms	Targets
TN1433	Batatasin III		FAK , Others , Akt
	Batatasin III inhibits cancer migration and invasion by suppressing epithelial to mesenchymal transition and FAK-AKT signals and possesses anti-cancer activities. Batatasin III has a long-term inhibitory effect on whole-...		FAK , Others , Akt
TQ0183	Narciclasine	Lycoricidinol	ROCK
	Narciclasine (Lycoricidinol), a natural product, modulates the Rho/Rho-kinase/LIM kinase/cofilin signaling pathway, greatly increasing GTPase RhoA activity.		ROCK
T8152	6-Demethoxytangeretin		MAPK , ALK
	6-Demethoxytangeretin is a citrus flavonoid isolated from Citrus depressa.		MAPK , ALK
T6677	Sophocarpine		ERK , p38 MAPK , NF-κB , TLR , COX , HER , JNK , STAT
	Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.		ERK , p38 MAPK , NF-κB , TLR , COX , HER , JNK , STAT
T0809	Dicoumarol	Dicumarol	Dehydrogenase , NADPH , PDK
	Dicoumarol (Dicumarol) is a hydroxycoumarin originally isolated from molding sweet-clover hay, with anticoagulant and vitamin K depletion activities. Dicoumarol is a competitive inhibitor of vitamin K epoxidereductase; t...		Dehydrogenase , NADPH , PDK
T2851	Daphnetin	7,8-Dihydroxycoumarin,Daphnetol	EGFR , PKA , PKC , Parasite , Autophagy
	Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM), and PKC (IC50: 25.01 μM), also exhibit anti-oxidant and anti-...		EGFR , PKA , PKC , Parasite , Autophagy
T5654	Musk ketone		Others
	Musk ketone can induce the growth repression and the apoptosis of cancer cells. Musk ketone increases activity of glutathione S-transferase and thus may prove to be useful cancer chemoprotectant.		Others
TN1828	Kahweol		Apoptosis , NF-κB , AMPK
	Kahweol has anticarcinogenic, anti-angiogenic,and anti-inflammatory activities, it can block the LPS-induced activation of NF-kappaB by preventing IkappaB degradation and inhibiting IkappaB kinase activity.		Apoptosis , NF-κB , AMPK
T2S2215	Crebanine		Apoptosis , Others , Akt
	1. Crebanine iv 5mg/kg can eonvert BaCl_2-induced arrhythmia into sinus rhythm in rats, and can significantly increase the tolerant dose of aconitine to produce ventrieular fibrillation(VF) and cardiac arrest (CA) in rat...		Apoptosis , Others , Akt
T4S1796	Heterophyllin B		PI3K
	Heterophyllin B effectively suppresses the adhesion and invasion of the human esophageal carcinoma cells by mediating the PI3K/AKT/β-catenin pathways and regulating the expression levels of adhesion- and invasion-associa...		PI3K
TN1557	Decursinol angelate		ERK , VEGFR , PKC , JNK
	Decursinol angelate has anti-tumor, anti-inflammatory, anti-oxidant, and hepatoprotective activities, it inhibits VEGF-induced angiogenesis via suppression of the VEGFR-2-signaling pathway; it also suppresses invasion an...		ERK , VEGFR , PKC , JNK
T5796	Plantainoside D	Isoplantamajoside	RAAS , PKC
	Plantainoside D (Isoplantamajoside) shows potent antioxidative effects as those of ascorbic acid, it shows angiotensin-converting enzyme (ACE) inhibitory inhibitory activity in vitro with the IC(50) value of 2.17 mM, it ...		RAAS , PKC
TMS1743	Salvigenin		MAO , Autophagy , ROS Kinase
	Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.		MAO , Autophagy , ROS Kinase
T2836	Isorhamnetin	3-methylquercetin,3'-Methylquercetin,Isorhamnetol,3'-Methoxyquercetin	MEK , PI3K , Endogenous Metabolite
	Isorhamnetin (3-methylquercetin) is the methylated metabolite of quercetin. Quercetin is an important dietary flavonoid with in vitro antioxidant activity. Isorhamnetin prevents endothelial cell injuries from oxidized LD...		MEK , PI3K , Endogenous Metabolite
T3889	Platycodin D		Prostaglandin Receptor , AMPK
	Platycodin D may stimulate TNF-α synthesis or inhibit degradation of TNF-α mRNA. Platycodin D (10/30 μM) suppresses prostaglandin E2 production in rat peritoneal macrophages stimulated by the protein kinase C activator 1...		Prostaglandin Receptor , AMPK
TN1100	Nepodin		transporter , COX , AMPK , Parasite
	Nepodin has antimalarial, and anti-inflammatory activities, it shows significant cyclooxygenase (COX) inhibitory activity. Nepodin has an antidiabetic effect, which is at least partly mediated by stimulation of GLUT4 tra...		transporter , COX , AMPK , Parasite
TN1299	Desmethylglycitein	6,7,4'-Trihydroxyisoflavone	PI3K , CDK , PKC
	Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which has antioxidant, and anti-cancer activities.		PI3K , CDK , PKC
T4672	Brevilin A		Apoptosis , Anti-infection , JAK , STAT , Autophagy
	Brevilin A is a sesquiterpene lactone isolated from Centipeda minima, inhibits janus kinase activity and blocks STAT3 signaling in cancer cells with anti-tumor activity. Brevilin A is a selective inhibitor of JAK-STAT si...		Apoptosis , Anti-infection , JAK , STAT , Autophagy
T5771	Hypocrellin A		Antibacterial , PKC , Parasite
	Hypocrellin A is PKC inhibitor, has light-induced antitumor,antifungal and antiviral activities, it also exerts immunomodulatory effects on MHC-restricted presentation of antigen.		Antibacterial , PKC , Parasite
T2798	Esculetin	Aesculetin,Cichorigenin	Lipoxygenase , Akt , PI3K
	Esculetin (Cichorigenin) is a coumarin derivative from various natural plant products with various biological and pharmaceutical properties including anti-edema, anti-inflammatory and anti-tumour effects. It inhibits lip...		Lipoxygenase , Akt , PI3K
T7190	Actein		Apoptosis , Akt , JNK , Autophagy
	Actein has a stimulatory effect on osteoblastic bone formation or has potential activity against osteoporosis, it also can prevent oxidative damage to osteoblasts in osteoporotic patients. Actein's ability to pathways in...		Apoptosis , Akt , JNK , Autophagy
T2746	Sophocarpine monohydrate	Sophocarpine	Apoptosis , Influenza Virus , Akt , PI3K , AMPK , Autophagy
	Sophocarpine monohydrate, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.		Apoptosis , Influenza Virus , Akt , PI3K , AMPK , Autophagy
TMS2181	Trans-Zeatin	(E)-Zeatin	ERK , MEK , Endogenous Metabolite
	trans-Zeatin ((E)-Zeatin) is the member of the plant growth hormone family known as cytokinins, which regulate cell division, development, and nutrient processing.		ERK , MEK , Endogenous Metabolite
T6S1302	Carnosol		Nrf2 , Endogenous Metabolite , S6 Kinase
	Carnosol is an Nrf2 activator, increasing Nrf2 levels and promoting heme oxygenase 1 (HMOX1) expression. It is a ribosomal S6 kinase (RSK2) inhibitor and can be used in gastric cancer-related research with an IC50 value ...		Nrf2 , Endogenous Metabolite , S6 Kinase
TN1134	Euscaphic acid		Apoptosis , LDL , PI3K , DNA/RNA Synthesis , NO Synthase , Prostaglandin Receptor
	Euscaphic acid has anti-diabetic, and anti-inflammatory activities, it inhibits LPS-induced inflammatory responses by interference with the clustering of TRAF6 with IRAK1 and TAK1, resulting in blocking the activation of...
T1711	Harmine	Telepathine	MAO , 5-HT Receptor , DYRK
	Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.		MAO , 5-HT Receptor , DYRK
T4S0498	Glaucocalyxin A	Wangzaozin B,Leukamenin F	Apoptosis , Akt , Caspase , PI3K
	1. Glaucocalyxin A (Leukamenin F)-SBE-β-CD could be useful with a better solubility and sustained function in drug delivery. 2. Glaucocalyxin A activates caspase-3, decreases BAD phosphorylation, and reduces the expressi...		Apoptosis , Akt , Caspase , PI3K
TN1405	Arnicolide D		Akt , Caspase , PI3K , STAT , mTOR
	Arnicolide D is a sesquiterpene lactone. Arnicolide D isolates from Centipeda minima. Arnicolide D modulates the cell cycle, activates the caspase signaling pathway and inhibits the PI3K/AKT/mTOR and STAT3 signaling path...		Akt , Caspase , PI3K , STAT , mTOR
T7327	7-Methoxyisoflavone		AMPK
	7-Methoxyisoflavone is an activator of adenosine monophosphate-activated protein kinase (AMPK).		AMPK
T3836	Eudesmin		MAPK , S6 Kinase
	Eudesmin shows antiinflammatory, neuritogenic, anticonvulsant and sedative effects, the mechanism of eudesmin may be related to up-regulation of GABAA and GAD65 expressions, and anti-apoptosis of neuron the in brain.50 m...		MAPK , S6 Kinase
T5S1467	Cucurbitacin E		CDK , Autophagy
	Cucurbitacin E is a natural product isolated from the climbing stem of Cucumic melo L. It significantly suppresses the activity of the cyclin B1/CDC2 complex.Cucurbitacin E has prevention of neurodegeneration, it has pot...		CDK , Autophagy
T3826	Polygalasaponin F		NF-κB , TLR , Akt , PI3K
	Polygalasaponin F has anti-neuroinflammatory activity, can inhibit the release of inflammatory cytokines TNF-α and NO induced by lipopolysaccharides (LPS) and reduce the expression of inducible nitric oxide synthases. Po...		NF-κB , TLR , Akt , PI3K
T5S0761	Nitidine chloride		Apoptosis , ERK , FAK , p38 MAPK , NF-κB , Topoisomerase , STAT , Parasite
	1. Nitidine chloride has inhibitory effects on various tumors, such as renal cancer , breast cancer. 2. Nitidine chloride inhibits the proliferation of SMMC-7721 cells in vitro in a time- and dose-dependent manner and id...
T2869	Emodin	Frangula emodin	SARS-CoV , Casein Kinase , Autophagy
	Emodin (Frangula emodin) is a naturally occurring anthraquinone present in the roots and barks of numerous plants; exerts antiproliferative effects in Y cells that are regulated by different signaling pathways.		SARS-CoV , Casein Kinase , Autophagy
T4S0800	Demethyleneberberine		P450 , NOS , NF-κB , HIF , AMPK
	Demethyleneberberine, which is composed of a potential antioxidant structure, could penetrate the membrane of mitochondria and accumulate in mitochondria either in vitro or in vivo.Demethyleneberberine suppresses CYP2E1,...		P450 , NOS , NF-κB , HIF , AMPK
T7030	Anemarsaponin B		p38 MAPK , NF-κB , MEK , COX , NO Synthase
	Anemarsaponin B has anti-inflammatory effect in LPS-treated RAW 264.7macrophages, the effect is associated with the inhibition of NF-κB transcriptional activity, possibly via the p38 MAP kinase pathway. Anemarsaponin B c...		p38 MAPK , NF-κB , MEK , COX , NO Synthase
T16324	Nimbolide		Apoptosis , NF-κB , CDK
	Nimbolide suppresses CDK4/CDK6 kinase activity. Nimbolide inhibits the NF-κB, Wnt, PI3K-Akt, MAPK, and JAK-STAT signaling pathways. Nimbolide causes apoptosis through the inactivation of NF-κB. Nimbolide is a triterpene ...		Apoptosis , NF-κB , CDK
T2811	Harmine hydrochloride	telepathine hydrochloride	5-HT Receptor , DYRK , GluR
	Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.		5-HT Receptor , DYRK , GluR
T3904	Gomisin J		Calcium Channel , AMPK
	Gomisin J is a natural product and have vasodilatory activity. Gomisin J suppresses lipid accumulation by regulating the expression of lipogenic and lipolytic enzymes and inflammatory molecules through activation of AMPK...		Calcium Channel , AMPK
T3881	Vaccarin		Integrin , Akt , PERK , AMPK
	Vaccarin is a major flavonoid glycoside in Vaccariae semen, its biotransformation pathways involves methylation, hydroxylation, glycosylation and deglycosylation.		Integrin , Akt , PERK , AMPK
TN4673	(+)-Nortrachelogenin	Wikstromol	Apoptosis , HIV Protease , PI3K , Antifection
	(+)-Nortrachelogenin is a lignan isolated from Wikstroemia indica C.A. Meyer (Thymelaeaceae). (+)-Nortrachelogenin possesses antileukemic activity.		Apoptosis , HIV Protease , PI3K , Antifection
TJS1779	Protosappanin A	PTA	NADPH-oxidase , IL Receptor , IκB/IKK , TNF , NF-κB , TLR , ROS , COX , HIV Protease , JAK , NO Synthase , STAT
	Protosappanin A (PTA) has anti-oxidative/nitrative activities on brain immune and neuroinflammation through regulation of CD14/TLR4-dependent IKK/IÎºB/NF-ÎºB inflammation signal pathway; it exerts anti-neuroinflammatory ...
T6630	Quercetin Dihydrate	Sophoretin	Apoptosis , PI3K
	Quercetin Dihydrate (Sophoretin) is a polyphenolic flavonoid that was found in a wide variety of plant-based foods, such as apples, onions, berries, and red wine. It is used for their nervous system and anticancer effect...		Apoptosis , PI3K
T5740	25(R,S)-Ruscogenin	(25RS)-Ruscogenin	Others , HIF
	25(R,S)-Ruscogenin is a natual product.		Others , HIF
T5497	AMAROGENTIN		Apoptosis , AMPK
	Amarogentin is mainly extracted from Swertia and Gentiana roots. It plays cemopreventive/therapeutic role during liver carcinogenesis through modulation of cell cycle and apoptosis		Apoptosis , AMPK
T2933	Wogonin	Vogonin	Apoptosis , Wnt/beta-catenin , CDK , Autophagy
	Wogonin (Vogonin) is a cell-permeable and orally available flavonoid that displays anti-inflammatory and anticancer properties.		Apoptosis , Wnt/beta-catenin , CDK , Autophagy
T1558	Resveratrol	trans-Resveratrol,SRT 501	Apoptosis , Mitophagy , IκB/IKK , Lipoxygenase , Sirtuin , COX , NADPH , DNA/RNA Synthesis , Nrf2 , Antibacterial , Antibiotic , Autophagy , Antifungal
	Resveratrol (SRT 501) is a polyphenolic natural product, a plant antitoxin with antioxidant and chemopreventive activities. Resveratrol has a wide range of targets including COX, SIRT, LOC, etc. Resveratrol induces autop...
T0167	Vinpocetine	RGH-4405,Ethyl apovincaminate	IκB/IKK , NF-κB , Sodium Channel , PDE
	Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).		IκB/IKK , NF-κB , Sodium Channel , PDE
T3122	Fangchinoline	Tetrandrine B,(+)-Limacine,Hanfangichin B,(+)-Fangchinoline	Apoptosis , FAK , HIV Protease , Autophagy
	Fangchinoline (Tetrandrine B) is extracted from Stephania tetrandra S. Moore.		Apoptosis , FAK , HIV Protease , Autophagy
T5S2017	Ingenol	(-)-Ingenol	PKC
	1. Ingenol ((-)-Ingenol) mebutate is an effective treatment for actinic keratosis. 2. Formulating novel derivatives from Ingenol esters may be an innovative approach to develop new lead compounds to reactivate latent HIV...		PKC
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Natural Products

Batatasin III

TN1433

Synonym:

Target: FAK, Others, Akt

Narciclasine

TQ0183

Synonym: Lycoricidinol

Target: ROCK

6-Demethoxytangeretin

Target: ERK, p38 MAPK, NF-κB, TLR, COX, HER, JNK, STAT

Dicoumarol

T0809

Synonym: Dicumarol

Target: Dehydrogenase, NADPH, PDK

Daphnetin

T2851

Synonym: 7,8-Dihydroxycoumarin,Daphnetol

Target: EGFR, PKA, PKC, Parasite, Autophagy

Target: Apoptosis, NF-κB, AMPK

Crebanine

T2S2215

Synonym:

Target: Apoptosis, Others, Akt

Target: ERK, VEGFR, PKC, JNK

Plantainoside D

T5796

Synonym: Isoplantamajoside

Target: MAO, Autophagy, ROS Kinase

Isorhamnetin

T2836

Synonym: 3-methylquercetin,3'-Methylquercetin,Isorhamnetol,3'-Methoxyquercetin

Target: MEK, PI3K, Endogenous Metabolite

Platycodin D

T3889

Synonym:

Target: Prostaglandin Receptor, AMPK

Nepodin

TN1100

Synonym:

Target: transporter, COX, AMPK, Parasite

Desmethylglycitein

TN1299

Synonym: 6,7,4'-Trihydroxyisoflavone

Target: PI3K, CDK, PKC

Brevilin A

T4672

Synonym:

Target: Apoptosis, Anti-infection, JAK, STAT, Autophagy

Hypocrellin A

T5771

Synonym:

Target: Antibacterial, PKC, Parasite

Esculetin

T2798

Synonym: Aesculetin,Cichorigenin

Target: Lipoxygenase, Akt, PI3K

Actein

T7190

Synonym:

Target: Apoptosis, Akt, JNK, Autophagy

Sophocarpine monohydrate

T2746

Synonym: Sophocarpine

Target: Apoptosis, Influenza Virus, Akt, PI3K, AMPK, Autophagy

trans-Zeatin

TMS2181

Synonym: (E)-Zeatin

Target: ERK, MEK, Endogenous Metabolite

Carnosol

T6S1302

Synonym:

Target: Nrf2, Endogenous Metabolite, S6 Kinase

Euscaphic acid

TN1134

Synonym:

Target: Apoptosis, LDL, PI3K, DNA/RNA Synthesis, NO Synthase, Prostaglandin Receptor

Harmine

T1711

Synonym: Telepathine

Target: MAO, 5-HT Receptor, DYRK

Glaucocalyxin A

T4S0498

Synonym: Wangzaozin B,Leukamenin F

Target: Apoptosis, Akt, Caspase, PI3K

Arnicolide D

TN1405

Synonym:

Target: Akt, Caspase, PI3K, STAT, mTOR

Target: MAPK, S6 Kinase

Cucurbitacin E

T5S1467

Synonym:

Target: CDK, Autophagy

Polygalasaponin F

T3826

Synonym:

Target: NF-κB, TLR, Akt, PI3K

Nitidine chloride

T5S0761

Synonym:

Target: Apoptosis, ERK, FAK, p38 MAPK, NF-κB, Topoisomerase, STAT, Parasite

Emodin

T2869

Synonym: Frangula emodin

Target: SARS-CoV, Casein Kinase, Autophagy

Demethyleneberberine

T4S0800

Synonym:

Target: P450, NOS, NF-κB, HIF, AMPK

anemarsaponin B

T7030

Synonym:

Target: p38 MAPK, NF-κB, MEK, COX, NO Synthase

Nimbolide

T16324

Synonym:

Target: Apoptosis, NF-κB, CDK

Harmine hydrochloride

T2811

Synonym: telepathine hydrochloride

Target: 5-HT Receptor, DYRK, GluR

Gomisin J

T3904

Synonym:

Target: Calcium Channel, AMPK

Vaccarin

T3881

Synonym:

Target: Integrin, Akt, PERK, AMPK

(+)-Nortrachelogenin

TN4673

Synonym: Wikstromol

Target: Apoptosis, HIV Protease, PI3K, Antifection

Protosappanin A

TJS1779

Synonym: PTA

Target: NADPH-oxidase, IL Receptor, IκB/IKK, TNF, NF-κB, TLR, ROS, COX, HIV Protease, JAK, NO Synthase, STAT

Quercetin Dihydrate

T6630

Synonym: Sophoretin

Target: Apoptosis, PI3K

25(R,S)-Ruscogenin

T5740

Synonym: (25RS)-Ruscogenin

Target: Apoptosis, AMPK

Wogonin

T2933

Synonym: Vogonin

Target: Apoptosis, Wnt/beta-catenin, CDK, Autophagy

Resveratrol

T1558

Synonym: trans-Resveratrol,SRT 501

Target: Apoptosis, Mitophagy, IκB/IKK, Lipoxygenase, Sirtuin, COX, NADPH, DNA/RNA Synthesis, Nrf2, Antibacterial, Antibiotic, Autophagy, Antifungal

Vinpocetine

T0167

Synonym: RGH-4405,Ethyl apovincaminate

Target: IκB/IKK, NF-κB, Sodium Channel, PDE

Fangchinoline

T3122

Synonym: Tetrandrine B,(+)-Limacine,Hanfangichin B,(+)-Fangchinoline

Target: Apoptosis, FAK, HIV Protease, Autophagy

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Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-04172	Adenylate Kinase 1 Protein, Rat, Recombinant (His)	Rat	E. coli
	The adenylate kinase (AK) isoforms network plays an important role in the intracellular energy transfer processes, the maintenance of energy homeostasis, and it is a major player in AMP metabolic signaling circuits in so...
TMPY-04412	Germinal Center Kinase/MAP4K2 Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	Mitogen-activated protein kinase kinase kinase kinase 2, also known as B lymphocyte serine/threonine-protein kinase, Germinal center kinase, MAPK/ERK kinase kinase kinase 2, MEK kinase kinase 2, Rab8-interacting protein,...
TMPH-00603	Cytidylate kinase Protein, E. coli, Recombinant (His & SUMO)	E. coli	E. coli
	ATP, dATP, and GTP are equally effective as phosphate donors. CMP and dCMP are the best phosphate acceptors.
TMPY-04432	Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant	Human	Baculovirus-Insect Cells
	SPHK1, also known as sphingosine Kinase 1, catalyzes the phosphorylation of sphingosine to form sphingosine-1-phosphate (S1P). S1P exhibits a broad spectrum of biological activities including cell proliferation, survival...
TMPY-04470	Adenylate Kinase 1 Protein, Human, Recombinant (His)	Human	E. coli
	The adenylate kinase (AK) isoforms network plays an important role in the intracellular energy transfer processes, the maintenance of energy homeostasis, and it is a major player in AMP metabolic signaling circuits in so...
TMPY-04403	NLK/Nemo Like Kinase Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	Nemo-like kinase contains 1 protein kinase domain and belongs to the protein kinase superfamily, CMGC Ser/Thr protein kinase family, and MAP kinase subfamily. It also contains a TQE activation loop motif in which autopho...
TMPY-04422	Casein Kinase 1 gamma 2 Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	Casein kinase I gamma 2 isoform (CSNK1G2), a member of the large casein kinase I (CKI) subfamily, protein kinase superfamily. It may affect the development of brain, and associate with vesicular trafficking and neurotran...
TMPY-04375	Casein Kinase 1 alpha Protein, Human, Recombinant (GST)	Human	Baculovirus-Insect Cells
	Casein kinase I isoform alpha, also known as CKI-alpha, CK1 and CSNK1A1, is a cytoplasm protein which belongs to theprotein kinase superfamily, CK1 Ser/Thr protein kinase family and casein kinase I subfamily. Casein k...
TMPY-04385	ZIP Kinase/DAPK3 Protein, Human, Recombinant (GST)	Human	Baculovirus-Insect Cells
	Death-associated protein kinase 3, also known as DAP kinase 3, ZIP-kinase, DAPK3 and ZIPK, is a nucleus and cytoplasm protein which belongs to theprotein kinase superfamily, CAMK Ser/Thr protein kinase family and DAP ...
TMPY-04431	Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	SPHK1, also known as sphingosine Kinase 1, catalyzes the phosphorylation of sphingosine to form sphingosine-1-phosphate (S1P). S1P exhibits a broad spectrum of biological activities including cell proliferation, survival...
TMPY-04356	GSK3B Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	GSK3B is a serine-threonine kinase, belonging to the glycogen synthase kinase subfamily. It Contains 1 protein kinase domain, and is expressed in the testis, thymus, prostate, and ovary and weakly expressed in the lung, ...
TMPY-04761	Creatine kinase B Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	CKB(Creatine kinase B type) contains 1 phosphagen kinase C-terminal domain and 1 phosphagen kinase N-terminal domain. It belongs to the ATP:guanido phosphotransferase family. CKB consists of a homodimer of two identical...
TMPH-03088	Arginine kinase/AK Protein, Penaeus monodon, Recombinant (His & SUMO)	Penaeus monodon	E. coli
	Arginine kinase/AK Protein, Penaeus monodon, Recombinant (His & SUMO) is expressed in E. coli.
TMPY-04406	Protein Kinase D2/PRKD2 Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	Serine/threonine-protein kinase D2, also known as PRKD2 and PKD2, is a cytoplasm and membrane protein that belongs to the protein kinase superfamily, CAMK Ser/Thr protein kinase family and PKD subfamily. PRKD2 / PKD2 is ...
TMPH-03503	Adenylate kinase Protein, Shigella flexneri, Recombinant (His & Myc & SUMO)	Shigella flexneri	E. coli
	Catalyzes the reversible transfer of the terminal phosphate group between ATP and AMP. Plays an important role in cellular energy homeostasis and in adenine nucleotide metabolism.
TMPY-04750	CSNK2A2 Protein, Human, Recombinant	Human	Baculovirus-Insect Cells
	Casein kinase II subunit alpha', also known as CSNK2A2 and CK2A2, is a member of the protein kinase superfamily, Ser/Thr protein kinase family and CK2 subfamily. Casein kinases are operationally defined by their prefer...
TMPY-00246	HER3/ERBB3 Protein, Rhesus, Recombinant	Rhesus	HEK293
	ErbB3, also known as Her3(human epidermal growth factor receptor3), is a member of the epidermal growth factor receptor (EGFR) family of receptor tyrosine kinases. This membrane-bound glycoprotein has a neuregulin bindin...
TMPY-04480	UMP-CMP kinase/CMPK1 Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	CMPK1 plays a key role in the maintenance of pyrimidine nucleotide pool profile and for the metabolism of pyrimidine analogs in cells. It catalyzes the phosphoryl transfer from ATP to UMP, CMP, and deoxy-CMP (dCMP), re...
TMPY-03024	HER3/ERBB3 Protein, Rat, Recombinant (His)	Rat	HEK293
	ErbB3, also known as Her3(human epidermal growth factor receptor3), is a member of the epidermal growth factor receptor (EGFR) family of receptor tyrosine kinases. This membrane-bound glycoprotein has a neuregulin bindin...
TMPY-04572	MKK4 Protein, Mouse, Recombinant (His & GST)	Mouse	Baculovirus-Insect Cells
	Dual specificity mitogen-activated protein kinase kinase 4, also known as MAP kinase kinase 4, MAPKK4, JNK-activating kinase 1, MAPK/ERK kinase 4, SAPK/ERK kinase 1, c-Jun N-terminal kinase kinase 1, JNKK, and MAP2K4, is...
TMPY-02813	ErbB4 Protein, Human, Rhesus, Recombinant (His)	Human,Rhesus	HEK293
	ERBB4 is a single-pass type I membrane protein with multiple cysteine rich domains, a transmembrane domain, a tyrosine kinase domain, a phosphotidylinositol-3 kinase binding site and a PDZ domain binding motif. ERBB4 is ...
TMPY-00548	HGFR/c-Met Protein, Cynomolgus, Rhesus, Recombinant (His)	Cynomolgus,Rhesus	HEK293
	Hepatocyte growth factor receptor (HGFR), also known as c-Met or mesenchymal-epithelial transition factor (MET), is a receptor tyrosine kinase (RTK) that is overexpressed and/or mutated in a variety of malignancies. HGFR...
TMPY-02477	HER3/ERBB3 Protein, Rhesus, Recombinant (His)	Rhesus	HEK293
	ErbB3, also known as Her3(human epidermal growth factor receptor3), is a member of the epidermal growth factor receptor (EGFR) family of receptor tyrosine kinases. This membrane-bound glycoprotein has a neuregulin bindin...
TMPY-04376	PLK1 Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	Serine / threonine-protein kinase PLK1 / PLK-1, also known as polo-like kinase 1 (PLK-1) or serine / threonine-protein kinase 13 (STPK13), Polo-like kinases (PLKs), is a family of four serine / threonine protein kinases ...
TMPY-01944	HER2/ERBB2 Protein, Rat, Recombinant (His)	Rat	HEK293
	Human epidermal growth factor receptor 2 (HER2), also known as ErbB2, NEU, and CD340, is a type I membrane glycoprotein and belongs to the epidermal growth factor (EGF) receptor family. HER2 protein cannot bind growth fa...
TMPY-00636	HER2/ERBB2 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293
	Human epidermal growth factor receptor 2 (HER2), also known as ErbB2, NEU, and CD340, is a type I membrane glycoprotein and belongs to the epidermal growth factor (EGF) receptor family. HER2 protein cannot bind growth fa...
TMPY-03719	HER2/ERBB2 Protein, Canine, Recombinant (His)	Canine	HEK293
	Human epidermal growth factor receptor 2 (HER2), also known as ErbB2, NEU, and CD340, is a type I membrane glycoprotein and belongs to the epidermal growth factor (EGF) receptor family. HER2 protein cannot bind growth fa...
TMPY-04548	CDK4 Protein, Human, Recombinant (GST)	Human	Baculovirus-Insect Cells
	CDK4 is a member of the Ser/Thr protein kinase family. It is highly similar to the gene products of S. cerevisiae cdc28 and S. pombe cdc2. It is a catalytic subunit of the protein kinase complex that is important for cel...
TMPJ-00412	VEGFR1/FLT-1 Protein, Human, Recombinant (hFc)	Human	Human Cells
	Human Vascular endothelial growth factor receptor 1(VEGFR-1, FLT-1) is a member of the the class III subfamily of receptor tyrosine kinases (RTKs) and Tyr protein kinase family and CSF-1/PDGF receptor subfamily. VEGFR-1 ...
TMPY-01601	AXL Protein, Human, Recombinant (His)	Human	HEK293
	Axl receptor tyrosine kinase, together with Tyro3 and Mer, constitute the TAM family of receptor tyrosine kinases. In the nervous system, Axl and its ligand Growth-arrest-specific protein 6 (Gas6) are expressed on multip...
TMPY-03215	FLT3 Ligand Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	FLT3L, also known as flt3 ligand, is a small molecule that acts as a growth factor that increases the number of immune cells by activating the hematopoietic progenitors. In vivo, FLT3L also induces the mobilization of th...
TMPY-06873	FLT3 Ligand Protein, Human, Recombinant	Human	E. coli
	FLT3L, also known as flt3 ligand, is a small molecule that acts as a growth factor that increases the number of immune cells by activating the hematopoietic progenitors. In vivo, FLT3L also induces the mobilization of th...
TMPY-03066	FLT3 Ligand Protein, Mouse, Recombinant (hFc)	Mouse	HEK293
	FLT3L, also known as flt3 ligand, is a small molecule that acts as a growth factor that increases the number of immune cells by activating the hematopoietic progenitors. In vivo, FLT3L also induces the mobilization of th...
TMPY-04649	ROR1 Protein, Human, Recombinant (His)	Human	HEK293

TMPY-01064	TIE2 Protein, Human, Recombinant (His)	Human	HEK293
	TEK, or TIE-2, is an endothelial cell-specific receptor tyrosine kinase (RTK) that is known as a functioning molecule of vascular endothelial cells. TEK comprises a subfamily of RTK with TIE, and these two receptors play...
TMPY-00930	TIE2 Protein, Human, Recombinant (His & hFc)	Human	HEK293
	TEK, or TIE-2, is an endothelial cell-specific receptor tyrosine kinase (RTK) that is known as a functioning molecule of vascular endothelial cells. TEK comprises a subfamily of RTK with TIE, and these two receptors play...
TMPY-05394	ROR2 Protein, Human, Recombinant (His)	Human	HEK293

TMPY-01247	FLT3 Protein, Human, Recombinant (T227M, His)	Human	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules which associating with th...
TMPY-00637	FLT1 Protein, Human, Recombinant (aa 1-328, His)	Human	HEK293
	Vascular endothelial growth factor receptor 1, also known as VEGFR-1, Fms-like tyrosine kinase 1, Tyrosine-protein kinase FRT, Tyrosine-protein kinase receptor FLT, Vascular permeability factor receptor and FLT1, is a si...
TMPY-02361	VEGFR2/KDR Protein, Human, Recombinant (His)	Human	HEK293
	VEGFR2 also called KDR or Flk-1, is identified as the receptor for VEGF and VEGFC and an early marker for endothelial cell progenitors, whose expression is restricted to endothelial cells in vivo. VEGFR2 was shown to be ...
TMPY-00882	Mer Protein, Human, Recombinant (His & hFc)	Human	HEK293
	Proto-oncogene tyrosine-protein kinase MER (MERTK) is a member of the MER/AXL/TYRO3 receptor kinase family and encodes a transmembrane protein with two fibronectin type-III domains, two Ig-like C2-type (immunoglobulin-li...
TMPY-01896	HGFR/c-Met Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Hepatocyte growth factor receptor (HGFR), also known as c-Met or mesenchymal-epithelial transition factor (MET), is a receptor tyrosine kinase (RTK) that is overexpressed and/or mutated in a variety of malignancies. HGFR...
TMPY-04330	Mer Protein, Human, Recombinant	Human	HEK293
	Proto-oncogene tyrosine-protein kinase MER (MERTK) is a member of the MER/AXL/TYRO3 receptor kinase family and encodes a transmembrane protein with two fibronectin type-III domains, two Ig-like C2-type (immunoglobulin-li...
TMPY-01936	VEGFR3/FLT4 Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Vascular endothelial growth factor receptor 3 (VEGFR3), also known as FLT-4, together with the other two members VEGFR1 (FLT-1) and VEGFR2 (KDR/Flk-1) are receptors for vascular endothelial growth factors (VEGF) and belo...
TMPJ-00778	HER2/ERBB2 Protein, Human, Recombinant (His)	Human	Human Cells
	Human epidermal growth factor receptor 2 (HER2) is a type of membrane glycoprotein, and belongs to the epidermal growth factor (EGF) receptor family. HER2 plays a key role in development, cell proliferation and different...
TMPY-04384	Src Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	Proto-oncogene tyrosine-protein kinase SRC is a hydrophobic protein belonging to the SRC family kinase including nine members that is a family of non-receptor tyrosine kinases. SRC protein may exist in different forms: C...
TMPY-02231	TrkB Protein, Mouse, Recombinant (His)	Mouse	HEK293
	TrkB receptor also known as TrkB tyrosine kinase or BDNF/NT-3 growth factors receptor or neurotrophic tyrosine kinase, receptor, type 2 (NTRK2) is a single transmembrane catalytic receptor with intracellular tyrosine kin...
TMPY-01296	HGFR/c-Met Protein, Human, Recombinant (His)	Human	HEK293
	Hepatocyte growth factor receptor (HGFR), also known as c-Met or mesenchymal-epithelial transition factor (MET), is a receptor tyrosine kinase (RTK) that is overexpressed and/or mutated in a variety of malignancies. HGFR...
TMPH-00904	Adenylate kinase 7 Protein, Human, Recombinant (His)	Human	Baculovirus
	Adenylate kinase 7 Protein, Human, Recombinant (His) is expressed in Baculovirus.
TMPY-01084	TrkA Protein, Human, Recombinant (His)	Human	HEK293
	TRKA is a member of the neurotrophic tyrosine kinase receptor (NTKR) family. It is a membrane-bound receptor that, upon neurotrophin binding, phosphorylates itself and members of the MAPK pathway. Isoform TrkA-III promot...
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Adenylate Kinase 1 Protein, Rat, Recombinant (His)

TMPY-04172

Species: Rat

Expression System: E. coli

Germinal Center Kinase/MAP4K2 Protein, Human, Recombinant (His & GST)

TMPY-04412

Species: Human

Expression System: Baculovirus-Insect Cells

Cytidylate kinase Protein, E. coli, Recombinant (His & SUMO)

TMPH-00603

Species: E. coli

Expression System: E. coli

Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant

TMPY-04432

Species: Human

Expression System: Baculovirus-Insect Cells

Adenylate Kinase 1 Protein, Human, Recombinant (His)

TMPY-04470

Species: Human

Expression System: E. coli

NLK/Nemo Like Kinase Protein, Human, Recombinant (His & GST)

TMPY-04403

Species: Human

Expression System: Baculovirus-Insect Cells

Casein Kinase 1 gamma 2 Protein, Human, Recombinant (His)

TMPY-04422

Species: Human

Expression System: Baculovirus-Insect Cells

Casein Kinase 1 alpha Protein, Human, Recombinant (GST)

TMPY-04375

Species: Human

Expression System: Baculovirus-Insect Cells

ZIP Kinase/DAPK3 Protein, Human, Recombinant (GST)

TMPY-04385

Species: Human

Expression System: Baculovirus-Insect Cells

Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant (His & GST)

TMPY-04431

Species: Human

Expression System: Baculovirus-Insect Cells

GSK3B Protein, Human, Recombinant (His)

TMPY-04356

Species: Human

Expression System: Baculovirus-Insect Cells

Creatine kinase B Protein, Human, Recombinant (His)

TMPY-04761

Species: Human

Expression System: Baculovirus-Insect Cells

Arginine kinase/AK Protein, Penaeus monodon, Recombinant (His & SUMO)

TMPH-03088

Species: Penaeus monodon

Expression System: E. coli

Protein Kinase D2/PRKD2 Protein, Human, Recombinant (His & GST)

TMPY-04406

Species: Human

Expression System: Baculovirus-Insect Cells

Adenylate kinase Protein, Shigella flexneri, Recombinant (His & Myc & SUMO)

TMPH-03503

Species: Shigella flexneri

Expression System: E. coli

CSNK2A2 Protein, Human, Recombinant

TMPY-04750

Species: Human

Expression System: Baculovirus-Insect Cells

HER3/ERBB3 Protein, Rhesus, Recombinant

TMPY-00246

Species: Rhesus

Expression System: HEK293

UMP-CMP kinase/CMPK1 Protein, Human, Recombinant (His)

TMPY-04480

Species: Human

Expression System: Baculovirus-Insect Cells

HER3/ERBB3 Protein, Rat, Recombinant (His)

TMPY-03024

Species: Rat

Expression System: HEK293

MKK4 Protein, Mouse, Recombinant (His & GST)

TMPY-04572

Species: Mouse

Expression System: Baculovirus-Insect Cells

ErbB4 Protein, Human, Rhesus, Recombinant (His)

TMPY-02813

Species: Human,Rhesus

Expression System: HEK293

HGFR/c-Met Protein, Cynomolgus, Rhesus, Recombinant (His)

TMPY-00548

Species: Cynomolgus,Rhesus

Expression System: HEK293

HER3/ERBB3 Protein, Rhesus, Recombinant (His)

TMPY-02477

Species: Rhesus

Expression System: HEK293

PLK1 Protein, Human, Recombinant (His)

TMPY-04376

Species: Human

Expression System: Baculovirus-Insect Cells

HER2/ERBB2 Protein, Rat, Recombinant (His)

TMPY-01944

Species: Rat

Expression System: HEK293

HER2/ERBB2 Protein, Cynomolgus, Recombinant (His)

TMPY-00636

Species: Cynomolgus

Expression System: HEK293

HER2/ERBB2 Protein, Canine, Recombinant (His)

TMPY-03719

Species: Canine

Expression System: HEK293

CDK4 Protein, Human, Recombinant (GST)

TMPY-04548

Species: Human

Expression System: Baculovirus-Insect Cells

VEGFR1/FLT-1 Protein, Human, Recombinant (hFc)

TMPJ-00412

Species: Human

Expression System: Human Cells

AXL Protein, Human, Recombinant (His)

TMPY-01601

Species: Human

Expression System: HEK293

FLT3 Ligand Protein, Human, Recombinant (His)

TMPY-03215

Species: Human

Expression System: Baculovirus-Insect Cells

FLT3 Ligand Protein, Human, Recombinant

TMPY-06873

Species: Human

Expression System: E. coli

FLT3 Ligand Protein, Mouse, Recombinant (hFc)

TMPY-03066

Species: Mouse

Expression System: HEK293

ROR1 Protein, Human, Recombinant (His)

TMPY-04649

Species: Human

Expression System: HEK293

TIE2 Protein, Human, Recombinant (His)

TMPY-01064

Species: Human

Expression System: HEK293

TIE2 Protein, Human, Recombinant (His & hFc)

TMPY-00930

Species: Human

Expression System: HEK293

ROR2 Protein, Human, Recombinant (His)

TMPY-05394

Species: Human

Expression System: HEK293

FLT3 Protein, Human, Recombinant (T227M, His)

TMPY-01247

Species: Human

Expression System: HEK293

FLT1 Protein, Human, Recombinant (aa 1-328, His)

TMPY-00637

Species: Human

Expression System: HEK293

VEGFR2/KDR Protein, Human, Recombinant (His)

TMPY-02361

Species: Human

Expression System: HEK293

Mer Protein, Human, Recombinant (His & hFc)

TMPY-00882

Species: Human

Expression System: HEK293

HGFR/c-Met Protein, Mouse, Recombinant (His)

TMPY-01896

Species: Mouse

Expression System: HEK293

Mer Protein, Human, Recombinant

TMPY-04330

Species: Human

Expression System: HEK293

VEGFR3/FLT4 Protein, Mouse, Recombinant (His)

TMPY-01936

Species: Mouse

Expression System: HEK293

HER2/ERBB2 Protein, Human, Recombinant (His)

TMPJ-00778

Species: Human

Expression System: Human Cells

Src Protein, Human, Recombinant (His & GST)

TMPY-04384

Species: Human

Expression System: Baculovirus-Insect Cells

TrkB Protein, Mouse, Recombinant (His)

TMPY-02231

Species: Mouse

Expression System: HEK293

HGFR/c-Met Protein, Human, Recombinant (His)

TMPY-01296

Species: Human

Expression System: HEK293

Adenylate kinase 7 Protein, Human, Recombinant (His)

TMPH-00904

Species: Human

Expression System: Baculovirus

TrkA Protein, Human, Recombinant (His)

TMPY-01084

Species: Human

Expression System: HEK293

--------- More ---------

Cat No.	Product Name
L1600	Kinase Inhibitor Library	2720 compounds
	A unique collection of 2720 kinase inhibitors/regulators for high throughput screening and high content screening for drug discovery in kinase related diseases;
L2200	Tyrosine Kinase Inhibitor Library	1033 compounds
	A unique collection of 1033 tyrosine kinase inhibitors for high throughput screening and high content screening for drug discovery in tyrosine kinase related diseases;
L1610	FDA-Approved Kinase Inhibitor Library	266 compounds
	A unique collection of 266 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening.
L1120	AMPK-Targeted Compound Library	80 compounds
	80 well-chosen unique AMPK-targeted small molecules；
L1300	PI3K-AKT-mTOR Compound Library	425 compounds
	A unique collection of 425 compounds targeting PI3K/Akt/mTOR signaling for research in PI3K/Akt/mTOR signaling, and drug discovery in diseases involved with PI3K/Akt/mTOR signaling;
L7700	Neural Regeneration Compound Library	529 compounds
	A unique collection of 149 neuroregeneration related compounds for high throughput and high content screening;
L2520	Glycometabolism Compound Library	708 compounds
	708 glycometabolism-related comounds, can be used for HTS and HCT;
L3800	NF-κB Signaling Compound Library	740 compounds
	A unique collection of 740 compounds targeting NF-κB signaling for high throughput screening and high content screening;
L1400	MAPK Inhibitor Library	367 compounds
	A unique collection of 367 compounds targeting MAPK signaling for drug discovery in MAPK related diseases;
L8000	Stem Cell Differentiation Compound Library	1213 compounds
	A unique collection of 1213 stem cell differentiation signaling targeted compounds for high throughput and high content screening;
L2191	Anti-Breast Cancer Compound Library	1965 compounds
	A unique collection of 1965 compounds with anti-breast cancer therapeutic activity or targeting breast cancer’s major signaling pathways, can be used for anti-breast cancer drug discovery and mechanism study；
L9410	Covalent Inhibitor Library	1949 compounds
	A unique collection of 1949 covalent Inhibitors and other molecules with common warheads like chloroacetyl，2-Chloropropionyl，Acryloyl，sulfonyl fluoride, alkyne，acrylamide, ketocarbonyl，disulfide bond, etc.