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PI-3065
Catalog No. T2083Cas No. 955977-50-1
PI-3065 is a novel potent and selective PI3K p110δ inhibitor.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $32 | In Stock | |
| 5 mg | $73 | In Stock | |
| 10 mg | $118 | In Stock | |
| 25 mg | $213 | In Stock | |
| 50 mg | $347 | In Stock | |
| 100 mg | $575 | In Stock | |
| 500 mg | $1,190 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | PI-3065 is a novel potent and selective PI3K p110δ inhibitor. |
| Targets&IC50 | p110δ:15 nM, p110β:1078 nM |
| In vitro | PI-3065 shows no inhibition on the growth of 4T1 cells, which do not expressing detectable levels of p110δ. [1] |
| Cell Research | Proliferation of 4T1 cells is assayed following a 4-h treatment with the indicated p110δ inhibitors, then washing and MTS staining are carried out after 48 h culture. (Only for Reference) |
| Alias | PI3065 |
| Molecular Weight | 506.64 |
| Formula | C27H31FN6OS |
| Cas No. | 955977-50-1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | DMSO: 1 mg/ml, Sonication is recommended.  |
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