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Ca2+ channel agonist 1

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Catalog No. T10659Cas No. 1402821-24-2

Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction.

Ca2+ channel agonist 1

Ca2+ channel agonist 1

🥰Excellent
Purity: 98.21%
Catalog No. T10659Cas No. 1402821-24-2
Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction.
Pack SizePriceAvailabilityQuantity
1 mg93 €In Stock
5 mg188 €In Stock
10 mg283 €In Stock
25 mg452 €In Stock
50 mg644 €In Stock
100 mg866 €In Stock
200 mg1.130 €In Stock
1 mL x 10 mM (in DMSO)217 €In Stock
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Purity:98.21%
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Product Introduction

Bioactivity
Description
Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction.
Targets&IC50
Ca2+ channel, N-type:14.23 μM (EC50), CDK2:3.34 μM (EC50)
In vitro
Ca2+ channel agonist 1 (Compound 13d) exhibits a ca. 2-fold increased agonism and a 22-fold decreased cdk2 kinase activity versus the standard, (R)-roscovitine.
Chemical Properties
Molecular Weight354.45
FormulaC19H26N6O
Cas No.1402821-24-2
SmilesCCCn1cnc2c(NCc3ccccc3)nc(N[C@H](CC)CO)nc12
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 45 mg/mL (126.96 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.8213 mL14.1064 mL28.2127 mL141.0636 mL
5 mM0.5643 mL2.8213 mL5.6425 mL28.2127 mL
10 mM0.2821 mL1.4106 mL2.8213 mL14.1064 mL
20 mM0.1411 mL0.7053 mL1.4106 mL7.0532 mL
50 mM0.0564 mL0.2821 mL0.5643 mL2.8213 mL
100 mM0.0282 mL0.1411 mL0.2821 mL1.4106 mL

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