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Eph inhibitor 2
🥰Excellent
Catalog No. T5451Cas No. 861249-59-4
Alias Ehp-inhibitor-1
Eph inhibitor 2 is an Eph family tyrosine kinase inhibitor targeting Eph receptors.
Eph inhibitor 2
🥰Excellent
Purity: 99.01%
Catalog No. T5451Alias Ehp-inhibitor-1Cas No. 861249-59-4
Eph inhibitor 2 is an Eph family tyrosine kinase inhibitor targeting Eph receptors.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $87 | In Stock | |
| 2 mg | $127 | In Stock | |
| 5 mg | $198 | In Stock | |
| 10 mg | $298 | In Stock | |
| 25 mg | $542 | In Stock | |
| 50 mg | $782 | In Stock | |
| 100 mg | $1,090 | In Stock | |
| 500 mg | $2,190 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $197 | In Stock |
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Dasatinib monohydrate (BMS-354825 Monohydrate) is an orally bioavailable synthetic small molecule-inhibitor of SRC-family protein-tyrosine kinases. Dasatinib monohydrate binds to and inhibits the growth-promoting activities of these kinases. Apparently, because of its less stringent binding affinity for the BCR-ABL kinase, Dasatinib monohydrate has been shown to overcome the resistance to imatinib of chronic myeloid leukemia (CML) cells harboring BCR-ABL kinase domain point mutations.
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ALW-II-49-7
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ALW-II-49-7 is a selective and potent inhibitor of EphB2 kinase, with an EC50 value of 40 nM in cell.
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AWL-II-38.3
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AWL-II-38.3 is a highly potent EphA3 inhibitor with potent kinase inhibitory activity against EphA3 but no significant cellular activity against Src family kinases or b-raf.
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JI-101
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Ehp-inhibitor-2
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Ehp-inhibitor-2 is an Eph family tyrosine kinase inhibitor targeting Eph receptors.
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Tivozanib
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123C4
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123C4 is a potent, selective, and competitive agonist of the receptor tyrosine kinase EPHA4 (Ki=0.65 μM)[1].
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NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
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ALW-II-41-27
Eph receptor tyrosine kinase inhibitor
T43441186206-79-0
ALW-II-41-27 (Eph receptor tyrosine kinase inhibitor), an Eph receptor tyrosine kinase inhibitor, is used for cancer therapy.
- $63
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Purity:99.01%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Eph inhibitor 2 is an Eph family tyrosine kinase inhibitor targeting Eph receptors. |
| Alias | Ehp-inhibitor-1 |
| Molecular Weight | 317.34 |
| Formula | C18H15N5O |
| Cas No. | 861249-59-4 |
| Smiles | NC=1N2C(=C(C=N2)C=3C=CC=NC3)N=CC1C4=CC(OC)=CC=C4 |
| Relative Density. | 1.34 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 32.5 mg/mL (102.41 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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