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PKC-theta inhibitor

Name: PKC-theta inhibitor
Brand: TargetMol
SKU: T5423
Rating: 4.5 (1 reviews)

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Catalog No. T5423Cas No. 736048-65-0

PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.

PKC-theta inhibitor

😃Good

Catalog No. T5423Cas No. 736048-65-0

PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.

Pack Size	Price	Availability
1 mg	$108	7-10 days
5 mg	$263	7-10 days
10 mg	$347	7-10 days
25 mg	$492	7-10 days
50 mg	$645	7-10 days
100 mg	$993	7-10 days
200 mg	$1,330	7-10 days
1 mL x 10 mM (in DMSO)	$288	7-10 days

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Product Introduction

Bioactivity

Description	PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.
Targets&IC50	PKCθ:12 nM

Chemical Properties

Molecular Weight	454.45
Formula	C₂₀H₂₅F₃N₆O₃
Cas No.	736048-65-0
Smiles	NCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
Relative Density.	1.356 g/cm3 (Predicted)

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 62.5 mg/mL (137.53 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.2005 mL	11.0023 mL	22.0046 mL	110.0231 mL
5 mM	0.4401 mL	2.2005 mL	4.4009 mL	22.0046 mL
10 mM	0.2200 mL	1.1002 mL	2.2005 mL	11.0023 mL
20 mM	0.1100 mL	0.5501 mL	1.1002 mL	5.5012 mL
50 mM	0.0440 mL	0.2200 mL	0.4401 mL	2.2005 mL
100 mM	0.0220 mL	0.1100 mL	0.2200 mL	1.1002 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc