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BIBF 1202
Catalog No. TQ0321Cas No. 894783-71-2
BIBF 1202 is a VEGFR2 kinase inhibitor (IC50 = 62 nM).
BIBF 1202
Catalog No. TQ0321Cas No. 894783-71-2
BIBF 1202 is a VEGFR2 kinase inhibitor (IC50 = 62 nM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $106 | In Stock | |
| 10 mg | $156 | In Stock | |
| 25 mg | $313 | In Stock | |
| 50 mg | $463 | In Stock | |
| 100 mg | $679 | In Stock | |
| 500 mg | $1,430 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $117 | In Stock |
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Purity:98.04%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | BIBF 1202 is a VEGFR2 kinase inhibitor (IC50: 62 nM). |
| Targets&IC50 | VEGFR2:62 nM |
| In vitro | The primary metabolic pathway for BIBF 1120 involves methyl ester cleavage to BIBF 1202, followed by glucuronidation of the free carboxyl group of BIBF 1202 to 1-O-acyl glucuronide [2]. |
| Molecular Weight | 525.6 |
| Formula | C30H31N5O4 |
| Cas No. | 894783-71-2 |
Storage & Solubility Information
| Storage | keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 40 mg/mL (76.1 mM) | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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